{"id":90224,"date":"2024-07-10T12:15:08","date_gmt":"2024-07-10T05:15:08","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=90224"},"modified":"2025-07-24T13:31:21","modified_gmt":"2025-07-24T06:31:21","slug":"olmac-5","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/olmac-5\/","title":{"rendered":"Olmac 5"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y, <\/b>d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/b><\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c Olmac 5<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi Macleods Pharmaceuticals Ltd – \u1ea4n \u0110\u1ed9, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-20555-17.<\/b><\/p>\n

Thu\u1ed1c Olmac 5 l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

Trong vi\u00ean n\u00e9n Olmac 5<\/b> bao g\u1ed3m c\u00e1c th\u00e0nh ph\u1ea7n nh\u01b0:<\/p>\n\n\n\n\n\n
Th\u00e0nh ph\u1ea7n<\/td>\nH\u00e0m l\u01b0\u1ee3ng<\/td>\n<\/tr>\n
Olanzapin<\/td>\n5mg<\/td>\n<\/tr>\n
T\u00e1 d\u01b0\u1ee3c<\/td>\nV\u1eeba \u0111\u1ee7<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n

D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim.<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: VN-20555-17.<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 3 v\u1ec9 x 10 vi\u00ean.<\/p>\n

Xu\u1ea5t x\u1ee9: \u1ea4n \u0110\u1ed9.<\/p>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Olmac 5<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

Olanzapin n\u1eb1m trong nh\u00f3m ch\u1ed1ng lo\u1ea1n th\u1ea7n th\u1ebf h\u1ec7 th\u1ee9 2. Thu\u1ed1c c\u00f3 th\u1ec3 ch\u1ed1ng lo\u1ea1n th\u1ea7n th\u00f4ng qua vi\u1ec7c ph\u1ed1i h\u1ee3p t\u00e1c \u0111\u1ed9ng \u0111\u1ed1i kh\u00e1ng 5-HT2 v\u00e0 dopamine. S\u1ef1 \u0111\u1ed1i kh\u00e1ng c\u1ee7a thu\u1ed1c v\u1edbi nh\u1eefng th\u1ee5 th\u1ec3 kh\u00e1c 2 th\u1ee5 th\u1ec3 n\u00eau tr\u00ean c\u00f3 th\u1ec3 gi\u1ea3i th\u00edch \u0111\u01b0\u1ee3c 1 s\u1ed1 t\u00e1c d\u1ee5ng tr\u1ecb li\u1ec7u v\u00e0 ph\u1ea3n \u1ee9ng ph\u1ee5 c\u1ee7a thu\u1ed1c.<\/p>\n

Ngo\u00e0i ra thu\u1ed1c c\u00f2n \u0111\u1ed1i kh\u00e1ng muscarinic t\u01b0\u01a1ng t\u1ef1 nh\u01b0 1 ch\u1ea5t \u0111\u1ed1i kh\u00e1ng cholinergic. C\u00f2n kh\u1ea3 n\u0103ng \u0111\u1ed1i kh\u00e1ng c\u1ee7a thu\u1ed1c tr\u00ean histamin H1 g\u00e2y ra t\u00ecnh tr\u1ea1ng bu\u1ed3n ng\u1ee7 khi s\u1eed d\u1ee5ng Olanzapin. Cu\u1ed1i c\u00f9ng thu\u1ed1c l\u00e0m t\u1ee5t huy\u1ebft \u00e1p th\u1ebf \u0111\u1ee9ng do vi\u1ec7c \u0111\u1ed1i kh\u00e1ng v\u1edbi alpha 1-adrenergic.<\/p>\n

\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

Thu\u1ed1c s\u1ebd \u0111\u01b0\u1ee3c h\u1ea5p thu t\u1ed1t sau khi d\u00f9ng vi\u00ean u\u1ed1ng, Cmax c\u00f3 sau 5-8 ti\u1ebfng. \u0110\u1ed3 \u0103n kh\u00f4ng g\u00e2y b\u1ea5t l\u1ee3i v\u1edbi vi\u1ec7c h\u1ea5p thu thu\u1ed1c.<\/p>\n

Kho\u1ea3ng 93% li\u1ec1u thu\u1ed1c v\u00e0o tu\u1ea7n ho\u00e0n g\u1eafn v\u00e0o protein, Vd g\u1ea7n 1000L.<\/p>\n

Thu\u1ed1c b\u1ecb chuy\u1ec3n h\u00f3a t\u1ea1i gan th\u00f4ng qua 2 qu\u00e1 tr\u00ecnh l\u00e0 li\u00ean h\u1ee3p v\u00e0 oxy h\u00f3a. 10-N-glucuronide l\u00e0 ch\u1ea5t chuy\u1ec3n h\u00f3a ch\u00ednh \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y, ch\u1ea5t chuy\u1ec3n h\u00f3a n\u00e0y kh\u00f4ng th\u1ec3 \u0111i qua m\u00e0ng n\u00e3o.<\/p>\n

Ngo\u00e0i ra c\u00f2n c\u00f3 2 ch\u1ea5t chuy\u1ec3n h\u00f3a l\u00e0 2-hydroxymethyl v\u00e0 N-desmethyl \u0111\u01b0\u1ee3c t\u1ea1o th\u00e0nh d\u01b0\u1edbi s\u1ef1 x\u00fac t\u00e1c c\u1ee7a CYP450. Hai ch\u1ea5t chuy\u1ec3n h\u00f3a c\u00f3 hi\u1ec7u qu\u1ea3 y\u1ebfu h\u01a1n nhi\u1ec1u so v\u1edbi Olanzapine.<\/p>\n

Th\u1eddi gian b\u00e1n h\u1ee7y kho\u1ea3ng 33 ti\u1ebfng v\u1edbi thanh th\u1ea3i huy\u1ebft t\u01b0\u01a1ng l\u00e0 26 l\u00edt m\u1ed7i gi\u1edd.<\/p>\n

Thu\u1ed1c Olmac 5 ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

Tr\u1ecb b\u1ec7nh cho ng\u01b0\u1eddi t\u00e2m th\u1ea7n ph\u00e2n li\u1ec7t hay c\u00f3 c\u01a1n h\u01b0ng c\u1ea3m l\u01b0\u1ee1ng c\u1ef1c.<\/p>\n

\"Thu\u1ed1c<\/a>
Thu\u1ed1c Olmac 5 \u0111i\u1ec1u tr\u1ecb t\u00e2m th\u1ea7n ph\u00e2n li\u1ec7t, h\u01b0ng c\u1ea3m<\/figcaption><\/figure>\n

Li\u1ec1u d\u00f9ng v\u00e0 c\u00e1ch d\u00f9ng thu\u1ed1c Olmac 5<\/h2>\n

Li\u1ec1u d\u00f9ng<\/h3>\n