{"id":57945,"date":"2023-11-20T09:38:54","date_gmt":"2023-11-20T02:38:54","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=57945"},"modified":"2025-07-24T13:44:17","modified_gmt":"2025-07-24T06:44:17","slug":"osart-20","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/osart-20\/","title":{"rendered":"Osart-20"},"content":{"rendered":"
Trong b\u00e0i vi\u1ebft n\u00e0y, D\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m Osart-20<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi Theon Pharmaceuticals Limited, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-21984-19<\/strong><\/p>\n M\u1ed7i vi\u00ean Osart-20<\/strong> c\u00f3 ch\u1ee9a:<\/p>\n D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim.<\/p>\n S\u0110K: VN-21984-19. Angiotensin I b\u1ecb th\u1ee7y ph\u00e2n nh\u1edd enzym chuy\u1ec3n d\u1ea1ng angiotensin (ACE) t\u1ea1o th\u00e0nh Angiotensin II c\u00f3 t\u00e1c d\u1ee5ng co m\u1ea1ch, k\u00edch th\u00edch tim, t\u0103ng t\u1ed5ng h\u1ee3p v\u00e0 gi\u1ea3i ph\u00f3ng aldosteron v\u00e0 t\u00e1i h\u1ea5p thu natri \u1edf th\u1eadn.<\/p>\n Olmesartan \u1ee9c ch\u1ebf ch\u1ecdn l\u1ecdc l\u00ean th\u1ee5 th\u1ec3 AT1 trong c\u01a1 tr\u01a1n m\u1ea1ch m\u00e1u, t\u1eeb \u0111\u00f3 \u1ee9c ch\u1ebf t\u00e1c d\u1ee5ng co m\u1ea1ch c\u1ee7a angiotensin II.<\/p>\n Kh\u00e1c v\u1edbi c\u00e1c ch\u1ea5t \u1ee9c ch\u1ebf ACE kh\u00e1c l\u00e0 \u1ee9c ch\u1ebf s\u1ef1 chuy\u1ec3n h\u00f3a c\u1ee7a bradykinin, th\u00ec olmesartan medoxomil kh\u00f4ng \u1ee9c ch\u1ebf ACE (kinase II) n\u00ean kh\u00f4ng \u1ea3nh h\u01b0\u1edfng \u0111\u1ebfn \u0111\u00e1p \u1ee9ng v\u1edbi bradykinin. Tuy nhi\u00ean ch\u01b0a th\u1ea5y s\u1ef1 kh\u00e1c bi\u1ec7t tr\u00ean l\u00e2m s\u00e0ng.<\/p>\n Trong qu\u00e1 tr\u00ecnh h\u1ea5p thu \u1edf \u0111\u01b0\u1eddng ti\u00eau h\u00f3a, Omesartan medoxomil chuy\u1ec3n h\u00f3a nhanh v\u00e0 ho\u00e0n to\u00e0n th\u00e0nh olmesartan nh\u1edd ph\u1ea3n \u1ee9ng th\u1ee7y ph\u00e2n ester.<\/p>\n Trong 3-5 ng\u00e0y, thu\u1ed1c \u0111\u1ea1t tr\u1ea1ng th\u00e1i \u1ed5n \u0111\u1ecbnh. Sinh kh\u1ea3 d\u1ee5ng tuy\u1ec7t \u0111\u1ed1i th\u1ea5p (26%) v\u00e0 kh\u00f4ng b\u1ecb \u1ea3nh h\u01b0\u1edfng b\u1edfi th\u1ee9c \u0103n. Sau khi u\u1ed1ng 1 – 2 gi\u1edd, thu\u1ed1c \u0111\u1ea1t n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng.<\/p>\n Th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 c\u1ee7a olmesartan x\u1ea5p x\u1ec9 171. 99% thu\u1ed1c li\u00ean k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng. Olmesartan kh\u00f4ng v\u00e0o \u0111\u01b0\u1ee3c t\u1ebf b\u00e0o h\u1ed3ng c\u1ea7u.<\/p>\n Thu\u1ed1c chuy\u1ec3n h\u00f3a nhanh v\u00e0 ho\u00e0n to\u00e0n trong qu\u00e1 tr\u00ecnh h\u1ea5p thu. \u0110\u1ed9 thanh th\u1ea3i huy\u1ebft t\u01b0\u01a1ng to\u00e0n ph\u1ea7n v\u00e0 c\u1ee7a th\u1eadn l\u1ea7n l\u01b0\u1ee3t l\u00e0 1,3 l\u00edt\/gi\u1edd v\u00e0 0,6 l\u00edt\/gi\u1edd.<\/p>\n C\u00f3 35% – 50% li\u1ec1u h\u1ea5p thu th\u1ea3i tr\u1eeb qua n\u01b0\u1edbc ti\u1ec3u, c\u00f2n l\u1ea1i qua ph\u00e2n v\u00e0 m\u1eadt.<\/p>\n Th\u1eddi gian b\u00e1n th\u1ea3i sau khi u\u1ed1ng trong kho\u1ea3ng 10 – 15 gi\u1edd.<\/p>\n D\u00f9ng \u0111\u01a1n \u0111\u1ed9c ho\u1eb7c ph\u1ed1i h\u1ee3p v\u1edbi c\u00e1c thu\u1ed1c h\u1ea1 \u00e1p kh\u00e1c trong \u0111i\u1ec1u tr\u1ecb t\u0103ng huy\u1ebft \u00e1p.<\/p>\nOsart-20 l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n
Th\u00e0nh ph\u1ea7n<\/h3>\n
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Tr\u00ecnh b\u00e0y<\/h3>\n
\nQuy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 3 v\u1ec9 x 10 vi\u00ean.
\nXu\u1ea5t x\u1ee9: \u1ea4n \u0110\u1ed9.<\/p>\nThu\u1ed1c Osart-20 c\u00f3 t\u00e1c d\u1ee5ng g\u00ec?<\/h2>\n
C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n
D\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n
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Thu\u1ed1c Osart-20 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n
Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Osart-20<\/h2>\n
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Kh\u00f4ng s\u1eed d\u1ee5ng thu\u1ed1c Osart-20 trong tr\u01b0\u1eddng h\u1ee3p n\u00e0o?<\/h2>\n
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L\u01b0u \u00fd \u0111\u1eb7c bi\u1ec7t trong qu\u00e1 tr\u00ecnh s\u1eed d\u1ee5ng thu\u1ed1c Osart-20<\/h2>\n
Th\u1eadn tr\u1ecdng<\/h3>\n
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T\u00e1c d\u1ee5ng ph\u1ee5<\/h3>\n