{"id":49108,"date":"2023-10-16T15:01:35","date_gmt":"2023-10-16T08:01:35","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=49108"},"modified":"2025-07-24T14:01:44","modified_gmt":"2025-07-24T07:01:44","slug":"nedaryl-4","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/nedaryl-4\/","title":{"rendered":"Nedaryl 4"},"content":{"rendered":"
Trong b\u00e0i vi\u1ebft n\u00e0y, d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m Nedaryl 4<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi C\u00f4ng ty c\u1ed5 ph\u1ea7n d\u01b0\u1ee3c Danapha. C\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VD-23440-15. Thu\u1ed1c \u0111\u01b0\u1ee3c d\u00f9ng \u1edf ng\u01b0\u1eddi m\u1eafc b\u1ec7nh Alzheimer \u0111\u1ec3 ch\u1ed1ng sa s\u00fat tr\u00ed tu\u1ec7.<\/b><\/p>\n Th\u00e0nh ph\u1ea7n c\u00f3 trong m\u1ed7i vi\u00ean n\u00e9n bao phim Nedaryl 4 g\u1ed3m c\u00f3:\u00a0<\/span><\/p>\n S\u0110K<\/span>:<\/b> VD-23440-15.<\/span><\/p>\n Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 1 v\u1ec9 x 14 vi\u00ean.<\/span><\/p>\n Xu\u1ea5t x\u1ee9: Vi\u1ec7t Nam.<\/span><\/p>\n Galantamine l\u00e0 ch\u1ea5t n\u1eb1m trong nh\u00f3m thu\u1ed1c \u1ee9c ch\u1ebf acetylcholinesterase. Galantamine g\u1eafn thu\u1eadn ngh\u1ecbch v\u00e0 l\u00e0m b\u1ea5t ho\u1ea1t acetylcholinesterase, do \u0111\u00f3 \u1ee9c ch\u1ebf th\u1ee7y ph\u00e2n acetylcholin, l\u00e0m t\u0103ng n\u1ed3ng \u0111\u1ed9 acetylcholin t\u1ea1i synap cholinergic. Ngo\u00e0i ra Galantamine c\u00f2n l\u00e0m t\u0103ng ho\u1ea1t t\u00ednh c\u1ee7a acetylcholin tr\u00ean th\u1ee5 th\u1ec3 nicotinic. S\u1ef1 thi\u1ebfu h\u1ee5t acetylcholin \u1edf v\u1ecf n\u00e3o, nh\u00e2n tr\u00e1m v\u00e0 h\u1ea3i m\u00e3 \u0111\u01b0\u1ee3c coi l\u00e0 m\u1ed9t trong nh\u1eefng \u0111\u1eb7c \u0111i\u1ec3m sinh l\u00fd b\u1ec7nh s\u1edbm c\u1ee7a b\u1ec7nh Alzheimer.<\/span><\/p>\n Galantamine \u0111\u01b0\u1ee3c \u0111\u00e1nh gi\u00e1 l\u00e0 h\u1ea5p thu nhanh v\u00e0 ho\u00e0n to\u00e0n. V\u1edbi sinh kh\u1ea3 d\u1ee5ng l\u00e0 90%. Galantamine sau khi v\u00e0o c\u01a1 th\u1ec3 s\u1ebd \u0111\u1ea1t n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh sau khi u\u1ed1ng kho\u1ea3ng 1 ti\u1ebfng.\u00a0\u00a0<\/span><\/p>\n Galantamine li\u00ean k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng kho\u1ea3ng 18%. Th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 trung b\u00ecnh c\u1ee7a thu\u1ed1c l\u00e0 175 l\u00edt.\u00a0<\/span><\/p>\n Galantamine chuy\u1ec3n h\u00f3a \u1edf gan th\u00f4ng qua cytochrom P450 v\u00e0 li\u00ean h\u1ee3p glucuronic.\u00a0<\/span><\/p>\n Kho\u1ea3ng 20% galantamine th\u1ea3i tr\u1eeb qua th\u1eadn d\u01b0\u1edbi d\u1ea1ng kh\u00f4ng \u0111\u1ed5i trong v\u00f2ng 24 gi\u1edd \u1edf ng\u01b0\u1eddi ch\u1ee9c n\u0103ng th\u1eadn b\u00ecnh th\u01b0\u1eddng, kho\u1ea3ng 20 – 25% \u0111\u1ed9 thanh th\u1ea3i to\u00e0n b\u1ed9 huy\u1ebft t\u01b0\u01a1ng l\u00e0 300ml\/ph\u00fat. N\u1eeda \u0111\u1eddi c\u1ee7a galantamine l\u00e0 5 – 7 gi\u1edd.<\/span><\/p>\n \u0110\u1ed1i v\u1edbi b\u1ec7nh nh\u00e2n b\u1ecb suy gan: Sau khi u\u1ed1ng 1 li\u1ec1u galantamine, \u0111\u1ed9 thanh th\u1ea3i galantamine b\u1ecb gi\u1ea3m kho\u1ea3ng 25% so v\u1edbi ng\u01b0\u1eddi b\u00ecnh th\u01b0\u1eddng.\u00a0<\/span><\/p>\n \u0110\u1ed1i v\u1edbi b\u1ec7nh nh\u00e2n b\u1ecb suy th\u1eadn: Sau m\u1ed9t li\u1ec1u duy nh\u1ea5t 8mg, AUC t\u0103ng kho\u1ea3ng 37% \u1edf ng\u01b0\u1eddi suy th\u1eadn v\u1eeba v\u00e0 67% \u1edf ng\u01b0\u1eddi suy th\u1eadn n\u1eb7ng so v\u1edbi ng\u01b0\u1eddi b\u00ecnh th\u01b0\u1eddng.\u00a0<\/span><\/p>\n \u0110\u1ed1i v\u1edbi b\u1ec7nh nh\u00e2n l\u00e0 ng\u01b0\u1eddi cao tu\u1ed5i: N\u1ed3ng \u0111\u1ed9 galantamine cao h\u01a1n so v\u1edbi ng\u01b0\u1eddi kh\u1ecfe m\u1ea1nh 30 – 40%.<\/span><\/p>\n Thu\u1ed1c Nedaryl 4 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh s\u1eed d\u1ee5ng trong \u0111i\u1ec1u tr\u1ecb ch\u1ee9ng sa s\u00fat tr\u00ed tu\u1ec7 t\u1eeb nh\u1eb9 \u0111\u1ebfn trung b\u00ecnh trong b\u1ec7nh Alzheimer.<\/span><\/p>\n Thu\u1ed1c Nedaryl 4 \u0111\u01b0\u1ee3c b\u00e0o ch\u1ebf d\u01b0\u1edbi d\u1ea1ng vi\u00ean n\u00e9n bao phim n\u00ean s\u1ebd \u0111\u01b0\u1ee3c s\u1eed d\u1ee5ng b\u1eb1ng \u0111\u01b0\u1eddng u\u1ed1ng.\u00a0<\/span><\/p>\n Thu\u1ed1c s\u1ebd \u0111\u01b0\u1ee3c u\u1ed1ng t\u1ed1t nh\u1ea5t v\u00e0o c\u00e1c b\u1eefa s\u00e1ng v\u00e0 b\u1eefa t\u1ed1i.<\/span><\/p>\nNedaryl 4 l\u00e0 thu\u1ed1c g\u00ec?<\/span><\/h2>\n
Th\u00e0nh ph\u1ea7n<\/span><\/h3>\n
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Tr\u00ecnh b\u00e0y<\/span><\/h3>\n
T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Nedaryl 4<\/span><\/h2>\n
\u0110\u1ed1i t\u01b0\u1ee3ng n\u00ean s\u1eed d\u1ee5ng Nedaryl 4<\/span><\/h2>\n
Li\u1ec1u d\u00f9ng – C\u00e1ch d\u00f9ng Nedaryl 4<\/span><\/h2>\n
C\u00e1ch d\u00f9ng<\/span><\/h3>\n
Li\u1ec1u d\u00f9ng<\/span><\/h3>\n