{"id":48604,"date":"2023-10-13T14:16:18","date_gmt":"2023-10-13T07:16:18","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=48604"},"modified":"2025-07-24T14:01:48","modified_gmt":"2025-07-24T07:01:48","slug":"ritozol-40mg","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/ritozol-40mg\/","title":{"rendered":"Ritozol 40mg"},"content":{"rendered":"
Trong b\u00e0i vi\u1ebft n\u00e0y, D\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c Ritozol 40mg<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi Bosch Pharmaceuticals (PVT) Ltd, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-16694-13<\/strong><\/p>\n M\u1ed7i vi\u00ean Ritozol 40mg<\/strong> c\u00f3 ch\u1ee9a:<\/p>\n D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean nang c\u1ee9ng (d\u1ea1ng h\u1ea1t c\u1ea3i bao tan trong ru\u1ed9t).<\/p>\n S\u0110K: VN-16694-13. Esomeprazole thu\u1ed9c nh\u00f3m PPI – thu\u1ed1c \u1ee9c ch\u1ebf b\u01a1m proton, l\u00e0 d\u1ea1ng \u0111\u1ed3ng ph\u00e2n S c\u1ee7a Omeprazole. Thu\u1ed1c \u0111\u1ea1t n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng sau khi u\u1ed1ng 1,5 gi\u1edd.<\/p>\n Li\u1ec1u t\u0103ng t\u1ec9 l\u1ec7 thu\u1eadn v\u1edbi n\u1ed3ng \u0111\u1ed9 thu\u1ed1c trong huy\u1ebft t\u01b0\u01a1ng, di\u1ec7n t\u00edch d\u01b0\u1edbi \u0111\u01b0\u1eddng cong (AUC) t\u0103ng 3 l\u1ea7n khi t\u0103ng li\u1ec1u t\u1eeb 20mg l\u00ean 40mg. U\u1ed1ng \u0111\u01a1n li\u1ec1u 40mg, sinh kh\u1ea3 d\u1ee5ng to\u00e0n th\u00e2n kho\u1ea3ng 64% so v\u1edbi li\u1ec1u 40mg l\u1eb7p l\u1ea1i h\u00e0ng ng\u00e0y th\u00ec sinh kh\u1ea3 d\u1ee5ng l\u00e0 90%.<\/p>\n Sau khi u\u1ed1ng \u0111\u01a1n li\u1ec1u Esomeprazole 40mg trong b\u1eefa \u0103n so v\u1edbi u\u1ed1ng l\u00fac \u0111\u00f3i, di\u1ec7n t\u00edch d\u01b0\u1edbi \u0111\u01b0\u1eddng cong gi\u1ea3m 43 \u2013 53%. Do \u0111\u00f3, Esomeprazole \u0111\u01b0\u1ee3c d\u00f9ng tr\u01b0\u1edbc \u0103n \u00edt nh\u1ea5t 1 gi\u1edd. Th\u1ee9c \u0103n l\u00e0m gi\u1ea3m v\u00e0 ch\u1eadm h\u1ea5p thu nh\u01b0ng kh\u00f4ng l\u00e0m thay \u0111\u1ed5i \u0111\u00e1ng k\u1ec3 t\u00e1c d\u1ee5ng gi\u1ea3m ti\u1ebft acid.<\/p>\n T\u1ef7 l\u1ec7 g\u1eafn v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng kh\u00e1 cao, kho\u1ea3ng 97%. Esomeprazole chuy\u1ec3n ho\u00e1 ho\u00e0n to\u00e0n qua h\u1ec7 th\u1ed1ng cytochrome P450 (CYP) th\u00e0nh ch\u1ea5t chuy\u1ec3n h\u00f3a thi\u1ebfu ho\u1ea1t t\u00ednh kh\u00e1ng ti\u1ebft.<\/p>\n Ph\u1ea7n l\u1edbn qu\u00e1 tr\u00ecnh chuy\u1ec3n h\u00f3a t\u1ea1o ra hydroxy v\u00e0 desmethyl \u0111\u01b0\u1ee3c th\u1ef1c hi\u1ec7n b\u1edfi isoenzyme CYP2C19. C\u00f2n l\u1ea1i t\u1ea1o th\u00e0nh ch\u1ea5t chuy\u1ec3n ho\u00e1 sulphone nh\u1edd v\u00e0o CYP3A4.<\/p>\n Trong huy\u1ebft t\u01b0\u01a1ng, th\u1eddi gian b\u00e1n th\u1ea3i ch\u00ednh trong kho\u1ea3ng 1 \u2013 1,5 gi\u1edd. D\u01b0\u1edbi 1% thu\u1ed1c \u1edf d\u1ea1ng kh\u00f4ng \u0111\u1ed5i \u0111\u01b0\u1ee3c \u0111\u00e0o th\u1ea3i trong n\u01b0\u1edbc ti\u1ec3u. Kho\u1ea3ng 80% li\u1ec1u thu\u1ed1c d\u01b0\u1edbi d\u1ea1ng ch\u1ea5t chuy\u1ec3n ho\u00e1 kh\u00f4ng ho\u1ea1t t\u00ednh \u0111\u01b0\u1ee3c \u0111\u00e0o th\u1ea3i qua n\u01b0\u1edbc ti\u1ec3u, ph\u1ea7n c\u00f2n l\u1ea1i \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y trong ph\u00e2n.<\/p>\n Thu\u1ed1c \u0111\u01b0\u1ee3c d\u00f9ng theo ch\u1ec9 \u0111\u1ecbnh c\u1ee7a th\u1ea7y thu\u1ed1c. Ng\u01b0\u1eddi l\u1edbn<\/p>\nRitozol 40mg l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n
Th\u00e0nh ph\u1ea7n<\/h3>\n
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Tr\u00ecnh b\u00e0y<\/h3>\n
\nQuy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 2 v\u1ec9 x 7 vi\u00ean.
\nXu\u1ea5t x\u1ee9: Pakistan.<\/p>\nThu\u1ed1c Ritozol 40mg c\u00f3 t\u00e1c d\u1ee5ng g\u00ec?<\/h2>\n
C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n
\nEsomeprazole t\u00e1c \u0111\u1ed9ng l\u00e0m gi\u1ea3m \u0111\u1ed9 acid trong d\u1ea1 d\u00e0y. C\u01a1 ch\u1ebf \u0111\u01b0\u1ee3c x\u00e1c \u0111\u1ecbnh l\u00e0 do ch\u1ea5t n\u00e0y \u1ee9c ch\u1ebf \u0111\u1eb7c hi\u1ec7u b\u01a1m proton H\/K – ATPase g\u1eafn \u1edf th\u00e0nh t\u1ebf b\u00e0o d\u1ea1 d\u00e0y – \u0111\u00e2y l\u00e0 giai \u0111o\u1ea1n cu\u1ed1i c\u00f9ng c\u1ee7a s\u1ef1 b\u00e0i ti\u1ebft acid.<\/p>\nD\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n
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\nTh\u1ec3 t\u00edch ph\u00e2n b\u1ed1 \u1ed5n \u0111\u1ecbnh kho\u1ea3ng 16l tr\u00ean ng\u01b0\u1eddi t\u00ecnh nguy\u1ec7n kho\u1ebb m\u1ea1nh.<\/p>\n\n
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Thu\u1ed1c Ritozol 40mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n
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<\/a>\n
Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Ritozol 40mg<\/h2>\n
C\u00e1ch d\u00f9ng<\/h3>\n
\nKh\u00f4ng b\u1ebb hay l\u00e0m v\u1ee1 vi\u00ean, nu\u1ed1t nguy\u00ean vi\u00ean v\u00e0 u\u1ed1ng tr\u01b0\u1edbc b\u1eefa \u0103n 1 gi\u1edd.<\/p>\nLi\u1ec1u d\u00f9ng<\/h3>\n