{"id":44324,"date":"2023-09-25T15:02:25","date_gmt":"2023-09-25T08:02:25","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=44324"},"modified":"2025-07-24T14:03:41","modified_gmt":"2025-07-24T07:03:41","slug":"clozapyl-25","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/clozapyl-25\/","title":{"rendered":"Clozapyl-25"},"content":{"rendered":"
Trong b\u00e0i vi\u1ebft n\u00e0y, d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c Clozapyl-25<\/a>\u00a0 \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi Th\u01b0\u01a1ng hi\u1ec7u Torrent Pharma (\u1ea4n \u0110\u1ed9) , c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-13897-11.<\/b><\/p>\n Trong m\u1ed7i vi\u00ean thu\u1ed1c Clozapyl-25<\/strong> c\u00f3 ch\u1ee9a th\u00e0nh ph\u1ea7n:<\/span><\/p>\n D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n<\/span><\/p>\n S\u0110K: VN-13897-11<\/span><\/p>\n Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 10 v\u1ec9 x 10 vi\u00ean.<\/span><\/p>\n Xu\u1ea5t x\u1ee9: \u1ea4n \u0110\u1ed9.<\/span><\/p>\n Clozapine c\u00f3 kh\u1ea3 n\u0103ng g\u1eafn k\u1ebft v\u00e0o receptor Dopamin v\u00e0 c\u00f3 t\u00e1c d\u1ee5ng kh\u00e1c v\u1edbi nh\u1eefng thu\u1ed1c \u1ee9c ch\u1ebf th\u1ea7n kinh \u0111i\u1ec3n h\u00ecnh h\u01a1n tr\u00ean c\u00e1c ph\u1ea3n \u1ee9ng ph\u1ee5 thu\u1ed9c Dopamin c\u1ee7a c\u01a1 th\u1ec3 n\u00ean \u0111\u01b0\u1ee3c x\u1ebfp v\u00e0o nh\u00f3m \u1ee9c ch\u1ebf t\u00e2m th\u1ea7n kh\u00f4ng \u0111i\u1ec3n h\u00ecnh.<\/span><\/p>\n Clozapine c\u00f3 \u00e1i l\u1ef1c cao v\u1edbi receptor D4 c\u1ee7a Dopamin, tuy nhi\u00ean l\u1ea1i ng\u0103n c\u1ea3n Dopamin li\u00ean k\u1ebft v\u1edbi c\u00e1c receptor D1, D2, D3, D5. Clozapine \u00edt c\u00f3 t\u00e1c d\u1ee5ng ph\u1ee5 \u1edf ngo\u1ea1i th\u00e1p, c\u00f3 t\u00e1c d\u1ee5ng nh\u01b0 m\u1ed9t ch\u1ea5t \u0111\u1ed1i kh\u00e1ng tr\u00ean c\u00e1c receptor Cholinergic, Serotonergic, Histaminergic, Adrenergic.<\/span><\/p>\n H\u1ea5p thu: D\u1ea1ng vi\u00ean n\u00e9n Clozapine<\/strong> c\u00f3 sinh kh\u1ea3 d\u1ee5ng t\u01b0\u01a1ng \u0111\u01b0\u01a1ng d\u1ea1ng dung d\u1ecbch, h\u1ea5p thu g\u1ea7n nh\u01b0 ho\u00e0n to\u00e0n b\u1eb1ng \u0111\u01b0\u1eddng u\u1ed1ng. N\u1ed3ng \u0111\u1ed9 \u0111\u1ea1t \u0111\u1ec9nh dao \u0111\u1ed9ng t\u1eeb 1 – 6 gi\u1edd trong huy\u1ebft t\u01b0\u01a1ng(Trung b\u00ecnh \u0111\u1ea1t \u0111\u1ec9nh sau kho\u1ea3ng 2,5 gi\u1edd).<\/span><\/p>\n Ph\u00e2n b\u1ed1: Clozapine ph\u00e2n b\u1ed1 r\u1ed9ng r\u00e3i trong c\u01a1 th\u1ec3, 97% Clozapine li\u00ean k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng.<\/span><\/p>\n Chuy\u1ec3n h\u00f3a: Clozapine \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a g\u1ea7n nh\u01b0 ho\u00e0n to\u00e0n tr\u01b0\u1edbc khi \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb. Ch\u1ea5t chuy\u1ec3n h\u00f3a d\u1ea1ng Hydroxyl h\u00f3a v\u00e0 N-oxy h\u00f3a kh\u00f4ng c\u00f3 t\u00e1c d\u1ee5ng, ch\u1ea5t chuy\u1ec3n h\u00f3a d\u1ea1ng Demethyl h\u00f3a ch\u1ec9 c\u00f2n r\u1ea5t \u00edt t\u00e1c d\u1ee5ng.<\/span><\/p>\n Th\u1ea3i tr\u1eeb: 50% qua n\u01b0\u1edbc ti\u1ec3u, 30% qua ph\u00e2n. Th\u1eddi gian b\u00e1n th\u1ea3i trung b\u00ecnh l\u00e0 8 gi\u1edd khi d\u00f9ng li\u1ec1u duy nh\u1ea5t 75mg Th\u1eddi gian b\u00e1n h\u1ee7y l\u00e0 12 gi\u1edd sau khi d\u00f9ng li\u1ec1u Clozapine \u1edf m\u1ee9c li\u1ec1u 100mgx2 l\u1ea7n\/ ng\u00e0y. Clozapine. \u0111\u01b0\u1ee3c \u0111\u00e0o th\u1ea3i ch\u1ee7 y\u1ebfu qua n\u01b0\u1edbc ti\u1ec3u v\u00e0 m\u1eadt.<\/span><\/p>\n Clozapyl-25 ch\u1ec9 \u0111\u1ecbnh trong \u0111i\u1ec1u tr\u1ecb t\u00e2m th\u1ea7n ph\u00e2n li\u1ec7t.<\/span><\/p>\nClozapyl-25 l\u00e0 thu\u1ed1c g\u00ec?<\/span><\/h2>\n
Th\u00e0nh ph\u1ea7n<\/span><\/h3>\n
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Tr\u00ecnh b\u00e0y<\/span><\/h3>\n
T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Clozapyl-25<\/span><\/h2>\n
C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng\u00a0<\/span><\/h3>\n
\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc\u00a0<\/span><\/h3>\n
Thu\u1ed1c Clozapyl-25 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/span><\/h2>\n
Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Clozapyl-25<\/span><\/h2>\n
Li\u1ec1u l\u01b0\u1ee3ng<\/span><\/h3>\n