{"id":44259,"date":"2023-09-25T11:24:46","date_gmt":"2023-09-25T04:24:46","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=44259"},"modified":"2025-07-24T14:03:41","modified_gmt":"2025-07-24T07:03:41","slug":"pregabakern-100-mg","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/pregabakern-100-mg\/","title":{"rendered":"Pregabakern 100mg"},"content":{"rendered":"
Trong b\u00e0i vi\u1ebft n\u00e0y, D\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c Pregabakern 100mg<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi KERN PHARMA S.L- T\u00e2y Ban Nha, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-22828-21<\/strong><\/p>\n M\u1ed7i vi\u00ean Pregabakern 100mg<\/strong> c\u00f3 ch\u1ee9a c\u00e1c th\u00e0nh ph\u1ea7n sau:<\/p>\n D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean nang c\u1ee9ng.<\/p>\n S\u0110K: VN-22828-21. Pregabalin thu\u1ed9c nh\u00f3m thu\u1ed1c ch\u1ed1ng \u0111\u1ed9ng kinh, l\u00e0 m\u1ed9t ch\u1ea5t t\u01b0\u01a1ng t\u1ef1 v\u1edbi acid gamma-aminobutyric [(S) -3- (aminomethyl) \u2013 5-methylhexanoic acid]. Khi u\u1ed1ng l\u00fac \u0111\u00f3i, Pregabalin \u0111\u01b0\u1ee3c h\u1ea5p thu nhanh. K\u1ec3 c\u1ea3 d\u00f9ng li\u1ec1u \u0111\u01a1n hay li\u1ec1u \u0111a, th\u00ec sau 1 gi\u1edd thu\u1ed1c \u0111\u1ea1t n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng. Sau khi d\u00f9ng \u0111\u01b0\u1eddng u\u1ed1ng, th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 bi\u1ec3u ki\u1ebfn c\u1ee7a pregabalin kho\u1ea3ng 0,56 L\/kg. Pregabalin kh\u00f4ng li\u00ean k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng.<\/p>\n Trong c\u01a1 th\u1ec3, Pregabalin \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a kh\u00f4ng \u0111\u00e1ng k\u1ec3. C\u00f3 kho\u1ea3ng 98% pregabalin \u1edf d\u1ea1ng ch\u01b0a chuy\u1ec3n h\u00f3a \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y trong n\u01b0\u1edbc ti\u1ec3u sau khi d\u00f9ng pregabalin \u0111\u00e1nh d\u1ea5u ph\u00f3ng x\u1ea1. Ch\u1ea5t chuy\u1ec3n h\u00f3a ch\u00ednh c\u1ee7a pregabalin l\u00e0 N-methylat \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y trong n\u01b0\u1edbc ti\u1ec3u. Nghi\u00ean c\u1ee9u ti\u1ec1n l\u00e2m s\u00e0ng cho th\u1ea5y kh\u00f4ng c\u00f3 s\u1ef1 bi\u1ebfn \u0111\u1ed5i \u0111\u1ed3ng ph\u00e2n pregabalin t\u1ea3 tuy\u1ec1n th\u00e0nh h\u1eefu tuy\u1ec1n.<\/p>\n Trung b\u00ecnh th\u1eddi gian b\u00e1n th\u1ea3i c\u1ee7a pregabalin l\u00e0 6,3 gi\u1edd. Pregabalin \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb ch\u1ee7 y\u1ebfu qua th\u1eadn. C\u1ea7n thi\u1ebft ph\u1ea3i \u0111i\u1ec1u ch\u1ec9nh li\u1ec1u tr\u00ean b\u1ec7nh nh\u00e2n suy gi\u1ea3m ch\u1ee9c n\u0103ng th\u1eadn v\u00e0 th\u1ea9m t\u00e1ch m\u00e1u.<\/p>\n D\u00f9ng thu\u1ed1c b\u1eb1ng \u0111\u01b0\u1eddng u\u1ed1ng. C\u00f3 th\u1ec3 u\u1ed1ng c\u00f9ng b\u1eefa \u0103n ho\u1eb7c kh\u00f4ng.<\/p>\n 1,5 – 6 vi\u00ean\/ng\u00e0y, chia th\u00e0nh 2-3 l\u1ea7n.<\/p>\n Kh\u1edfi \u0111\u1ea7u v\u1edbi li\u1ec1u 1,5 vi\u00ean\/ng\u00e0y, chia 2-3 l\u1ea7n. C\u00f3 th\u1ec3 t\u0103ng l\u00ean 3 vi\u00ean\/ng\u00e0y sau 3-7 ng\u00e0y d\u1ef1a v\u00e0o \u0111\u00e1p \u1ee9ng v\u00e0 kh\u1ea3 n\u0103ng dung n\u1ea1p c\u1ee7a b\u1ec7nh nh\u00e2n. N\u1ebfu c\u1ea7n t\u0103ng li\u1ec1u \u0111\u1ebfn t\u1ed1i \u0111a 6 vi\u00ean\/ng\u00e0y sau 7 ng\u00e0y.<\/p>\n Kh\u1edfi \u0111\u1ea7u v\u1edbi li\u1ec1u 1,5 vi\u00ean\/ng\u00e0y, chia 2-3 l\u1ea7n. C\u00f3 th\u1ec3 t\u0103ng l\u00ean 3 vi\u00ean\/ng\u00e0y sau 1 tu\u1ea7n d\u1ef1a v\u00e0o \u0111\u00e1p \u1ee9ng v\u00e0 kh\u1ea3 n\u0103ng dung n\u1ea1p c\u1ee7a b\u1ec7nh nh\u00e2n. N\u1ebfu c\u1ea7n t\u0103ng li\u1ec1u \u0111\u1ebfn t\u1ed1i \u0111a 6 vi\u00ean\/ng\u00e0y sau 1 tu\u1ea7n n\u1eefa.<\/p>\n Li\u1ec1u d\u00f9ng t\u1eeb 1,5-6 vi\u00ean\/ng\u00e0y, chia 2-3 l\u1ea7n.Pregabakern 100mg l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n
Th\u00e0nh ph\u1ea7n<\/h3>\n
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\n Ho\u1ea1t ch\u1ea5t<\/td>\n T\u00e1 d\u01b0\u1ee3c<\/td>\n V\u1ecf nang<\/td>\n M\u1ef1c in m\u00e0u \u0111en<\/td>\n<\/tr>\n \n Pregabalin 100 mg<\/td>\n Lactose monohydrat (phun s\u1ea5y), talc, tinh b\u1ed9t ng\u00f4.<\/td>\n Gelatin, oxit s\u1eaft \u0111\u1ecf, titanium dioxide.<\/td>\n Shellac, dung d\u1ecbch amoniac \u0111\u1eadm \u0111\u1eb7c, kali hydroxid, propylen glycol, oxid s\u1eaft \u0111en t\u1ed5ng h\u1ee3p.<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n Tr\u00ecnh b\u00e0y<\/h3>\n
\nQuy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 6 v\u1ec9 x 14 vi\u00ean.
\nXu\u1ea5t x\u1ee9: T\u00e2y Ban Nha.<\/p>\nT\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Pregabakern 100mg<\/h2>\n
C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n
\nPregabalin t\u00e1c \u0111\u1ed9ng v\u00e0o h\u1ec7 th\u1ed1ng th\u1ea7n kinh trung \u01b0\u01a1ng b\u1eb1ng c\u00e1ch g\u1eafn v\u1edbi m\u1ed9t nh\u00f3m ph\u1ee5 c\u1ee7a d\u00f2ng canxi mang \u0111i\u1ec7n.<\/p>\n\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n
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\nSinh kh\u1ea3 d\u1ee5ng \u0111\u01b0\u1eddng u\u1ed1ng kh\u00e1 cao (kho\u1ea3ng 90%) v\u00e0 ph\u1ee5 thu\u1ed9c li\u1ec1u d\u00f9ng. N\u1ed3ng \u0111\u1ed9 thu\u1ed1c \u1ed5n \u0111\u1ecbnh trong 24-48 gi\u1edd khi d\u00f9ng nh\u1eafc l\u1ea1i. Khi d\u00f9ng c\u00f9ng th\u1ee9c \u0103n s\u1ef1 h\u1ea5p thu c\u1ee7a thu\u1ed1c gi\u1ea3m th\u1ec3 hi\u1ec7n: Cmax gi\u1ea3m kho\u1ea3ng 25-30% v\u00e0 tmax k\u00e9o d\u00e0i kho\u1ea3ng 2,5 gi\u1edd. Tuy nhi\u00ean, kh\u00f4ng \u1ea3nh h\u01b0\u1edfng \u0111\u00e1ng k\u1ec3 \u0111\u1ebfn m\u1ee9c \u0111\u1ed9 h\u1ea5p thu pregabalin.<\/p>\n\n
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\n \u0110\u1ed1i t\u01b0\u1ee3ng<\/td>\n D\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/td>\n<\/tr>\n \n Suy th\u1eadn<\/td>\n Thanh th\u1ea3i creatinin t\u1ec9 l\u1ec7 thu\u1eadn v\u1edbi thanh th\u1ea3i pregabalin. Pregabalin \u0111\u01b0\u1ee3c lo\u1ea1i b\u1ecf kh\u1ecfi huy\u1ebft t\u01b0\u01a1ng nh\u1edd th\u1ea9m t\u00e1ch m\u00e1u. Pregabalin ch\u1ee7 y\u1ebfu \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb qua th\u1eadn, n\u00ean b\u1ec7nh nh\u00e2n suy th\u1eadn c\u1ea7n gi\u1ea3m li\u1ec1u v\u00e0 b\u1ec7nh nh\u00e2n th\u1ea9m t\u00e1ch m\u00e1u c\u1ea7n ph\u1ea3i b\u1ed5 sung li\u1ec1u.<\/td>\n<\/tr>\n \n Suy gan<\/td>\n Ch\u01b0a c\u00f3 nhi\u1ec1u c\u00e1c nghi\u00ean c\u1ee9u tr\u00ean b\u1ec7nh nh\u00e2n suy gan. Kh\u00f4ng c\u00f3 s\u1ef1 thay \u0111\u1ed5i \u0111\u00e1ng k\u1ec3 v\u1ec1 n\u1ed3ng \u0111\u1ed9 huy\u1ebft t\u01b0\u01a1ng \u1edf b\u1ec7nh nh\u00e2n n\u00e0y.<\/td>\n<\/tr>\n \n Tr\u1ebb em<\/td>\n Nghi\u00ean c\u1ee9u tr\u00ean b\u1ec7nh nh\u00e2n nhi \u0111\u1ed9ng kinh, sau khi u\u1ed1ng Pregabalin l\u00fac \u0111\u00f3i 0,5-2 gi\u1edd th\u00ec thu\u1ed1c \u0111\u1ea1t n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng.
\nCmax v\u00e0 AUC c\u1ee7a pregabalin t\u0103ng t\u01b0\u01a1ng \u1ee9ng v\u1edbi li\u1ec1u t\u0103ng l\u00ean. B\u1ec7nh nh\u00e2n nhi d\u01b0\u1edbi 30 kg AUC th\u1ea5p h\u01a1n 30%.
\nTh\u1eddi gian b\u00e1n th\u1ea3i kho\u1ea3ng 3-4 gi\u1edd \u1edf b\u1ec7nh nh\u00e2n nhi d\u01b0\u1edbi 6 tu\u1ed5i v\u00e0 t\u1eeb 4-6 gi\u1edd \u1edf tr\u1ebb t\u1eeb 7 tu\u1ed5i tr\u1edf l\u00ean.
\nCh\u01b0a nghi\u00ean c\u1ee9u d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc c\u1ee7a pregabalin \u1edf tr\u1ebb d\u01b0\u1edbi 3 th\u00e1ng tu\u1ed5i.<\/td>\n<\/tr>\n\n Ng\u01b0\u1eddi gi\u00e0<\/td>\n Tu\u1ed5i c\u00e0ng t\u0103ng th\u00ec \u0111\u1ed9 thanh th\u1ea3i c\u1ee7a pregabalin c\u00e0ng c\u00f3 xu h\u01b0\u1edbng gi\u1ea3m. Ng\u01b0\u1eddi gi\u00e0 c\u00f3 t\u1ed5n th\u01b0\u01a1ng ch\u1ee9c n\u0103ng th\u1eadn c\u1ea7n gi\u1ea3m li\u1ec1u.<\/td>\n<\/tr>\n \n Ph\u1ee5 n\u1eef cho con b\u00fa<\/td>\n D\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc pregabalin \u00edt ho\u1eb7c kh\u00f4ng b\u1ecb \u1ea3nh h\u01b0\u1edfng khi cho con b\u00fa. Kho\u1ea3ng 76% pregabalin b\u00e0i ti\u1ebft v\u00e0o s\u1eefa m\u1eb9 so v\u1edbi n\u1ed3ng \u0111\u1ed9 trong huy\u1ebft t\u01b0\u01a1ng.
\nKhi ng\u01b0\u1eddi m\u1eb9 d\u00f9ng pregabalin 300 mg\/ng\u00e0y ho\u1eb7c t\u1ed1i \u0111a 600 mg\/ng\u00e0y th\u00ec li\u1ec1u l\u01b0\u1ee3ng tr\u1ebb s\u01a1 sinh \u01b0\u1edbc t\u00ednh nh\u1eadn \u0111\u01b0\u1ee3c t\u1eeb s\u1eefa m\u1eb9 l\u00e0 0,31 ho\u1eb7c 0.62 mg\/kg\/ng\u00e0y.<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\nThu\u1ed1c Pregabakern 100mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n
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Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Pregabakern 100mg<\/h2>\n
C\u00e1ch d\u00f9ng<\/h3>\n
Li\u1ec1u d\u00f9ng<\/h3>\n
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\nPregabalin c\u00f3 th\u1ec3 \u0111\u01b0\u1ee3c kh\u1edfi \u0111\u1ea7u v\u1edbi li\u1ec1u 1,5 vi\u00ean\/ ng\u00e0y. C\u00f3 th\u1ec3 t\u0103ng l\u00ean 3 vi\u00ean\/ng\u00e0y sau 1 tu\u1ea7n d\u1ef1a v\u00e0o \u0111\u00e1p \u1ee9ng v\u00e0 kh\u1ea3 n\u0103ng dung n\u1ea1p c\u1ee7a b\u1ec7nh nh\u00e2n. Tu\u1ea7n sau \u0111\u00f3, c\u00f3 th\u1ec3 t\u0103ng li\u1ec1u l\u00ean \u0111\u1ebfn 4,5 vi\u00ean\/ ng\u00e0y. N\u1ebfu c\u1ea7n t\u0103ng li\u1ec1u \u0111\u1ebfn t\u1ed1i \u0111a 6 vi\u00ean\/ng\u00e0y sau 1 tu\u1ea7n n\u1eefa.<\/p>\n\n