{"id":42408,"date":"2023-09-15T15:12:14","date_gmt":"2023-09-15T08:12:14","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=42408"},"modified":"2025-07-24T14:03:47","modified_gmt":"2025-07-24T07:03:47","slug":"thuoc-cales-20mg","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/thuoc-cales-20mg\/","title":{"rendered":"C.ales 20mg"},"content":{"rendered":"
Trong b\u00e0i vi\u1ebft n\u00e0y, d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c C.ales 20mg<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi C\u00f4ng ty C\u1ed5 ph\u1ea7n D\u01b0\u1ee3c ph\u1ea9m C\u1eedu Long, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VD-23519-15.<\/strong><\/p>\n Thu\u1ed1c C.ales 20mg c\u00f3 ch\u1ee9a th\u00e0nh ph\u1ea7n:<\/p>\n D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim.<\/p>\n S\u0110K: VD-23519-15 Thu\u1ed1c \u0111\u01b0\u1ee3c d\u00f9ng trong r\u1ed1i lo\u1ea1n c\u01b0\u01a1ng d\u01b0\u01a1ng. Guanosin Monophosphat v\u00f2ng (cGMP) b\u1ecb Tadalafil \u1ee9c ch\u1ebf ch\u1ecdn l\u1ecdc c\u00f3 h\u1ed3i ph\u1ee5c, \u0111\u1eb7c bi\u1ec7t l\u00e0 tr\u00ean PDE5. Trong \u0111\u00f3 PDE5 phosphodiesterase type 5) l\u00e0 enzyme \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y \u1edf c\u01a1 tr\u01a1n m\u1ea1ch m\u00e1u v\u00e0 t\u1ea1ng, c\u01a1 tr\u01a1n th\u1ec3 hang, c\u01a1 x\u01b0\u01a1ng, ti\u1ec3u c\u1ea7u, th\u1eadn,ti\u1ec3u n\u00e3o, ph\u1ed5i. Tadalafil t\u00e1c \u0111\u1ed9ng tr\u00ean PDE5 m\u1ea1nh h\u01a1n c\u00e1c Phosphodiesterase.<\/p>\n PDE1, PDE2, PDE4 v\u00e0 PDE7 l\u00e0 c\u00e1c enzym xu\u1ea5t hi\u1ec7n \u1edf n\u00e3o, tim, gan, m\u1ea1ch m\u00e1u, v\u00e0 nh\u1eefng c\u01a1 quan kh\u00e1c. PDE3 xu\u1ea5t hi\u1ec7n trong m\u1ea1ch m\u00e1u, tim. PDE6 l\u00e0 men xu\u1ea5t hi\u1ec7n trong v\u00f5ng m\u1ea1c. Tadalafil t\u00e1c \u0111\u1ed9ng tr\u00ean PDE5 m\u1ea1nh h\u01a1n PDE11A1 v\u00e0 PDE11A4 l\u1ea7n l\u01b0\u1ee3t l\u00e0 14 v\u00e0 40 l\u1ea7n. Trong \u0111\u00f3 PDE11A1 v\u00e0 PDE11A4 l\u00e0 hai trong s\u1ed1 4 h\u00ecnh th\u1ee9c \u0111\u01b0\u1ee3c bi\u1ebft c\u1ee7a PDE 11( \u0111\u00e2y l\u00e0 m\u1ed9t lo\u1ea1i men t\u00ecm th\u1ea5y trong tuy\u1ebfn ti\u1ec1n li\u1ec7t, c\u01a1 x\u01b0\u01a1ng, tinh ho\u00e0n v\u00e0 c\u00e1c m\u00f4 kh\u00e1c).<\/p>\n Tadalafil h\u1ea5p thu nhanh sau khi u\u1ed1ng. Sau 2 gi\u1edd u\u1ed1ng th\u00ec \u0111\u1ea1t \u0111\u01b0\u1ee3c n\u1ed3ng \u0111\u1ed9 t\u1ed1i \u0111a trong huy\u1ebft t\u01b0\u01a1ng. C\u00f3 th\u1ec3 d\u00f9ng thu\u1ed1c trong ho\u1eb7c ngo\u00e0i b\u1eefa \u0103n v\u00ec l\u01b0\u1ee3ng th\u1ee9c \u0103n kh\u00f4ng l\u00e0m \u1ea3nh h\u01b0\u1edfng \u0111\u1ebfn t\u1ed1c \u0111\u1ed9 h\u1ea5p thu c\u1ee7a Tadalafil.<\/p>\n Th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 kho\u1ea3ng 63L. Tadalafil g\u1eafn v\u1edbi protein huy\u1ebft kho\u1ea3ng 94% v\u00e0 kh\u00f4ng b\u1ecb \u1ea3nh h\u01b0\u1edfng b\u1edfi ch\u1ee9c n\u0103ng c\u1ee7a th\u1eadn.<\/p>\n Tadalafil chuy\u1ec3n h\u00f3a ch\u1ee7 y\u1ebfu qua cytochrom P450 (CYP) v\u00e0 Methylcatechol Glucuronic l\u00e0 ch\u1ea5t chuy\u1ec3n h\u00f3a c\u00f3 ho\u1ea1t t\u00ednh.<\/p>\n Khi d\u00f9ng \u0111\u01b0\u1eddng u\u1ed1ng, \u0111\u1ed9 thanh th\u1ea3i c\u1ee7a Tadalafil kho\u1ea3ng 2,5 gi\u1edd. Th\u1eddi gian b\u00e1n h\u1ee7y b\u00ecnh th\u01b0\u1eddng l\u00e0 17,5 gi\u1edd. Thu\u1ed1c C.ales 20mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh d\u00f9ng trong c\u00e1c tr\u01b0\u1eddng h\u1ee3p sau:<\/p>\nC.ales 20mg l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n
Th\u00e0nh ph\u1ea7n<\/h3>\n
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Tr\u00ecnh b\u00e0y<\/h3>\n
\nQuy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 1 v\u1ec9 x 1 vi\u00ean.
\nXu\u1ea5t x\u1ee9: Vi\u1ec7t Nam.<\/p>\nT\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c C.ales 20mg?<\/h2>\n
C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n
\nNitric oxide s\u1ebd \u0111\u01b0\u1ee3c ph\u00f3ng th\u00edch t\u1ea1i ch\u1ed7 khi c\u00f3 k\u00edch th\u00edch t\u00ecnh d\u1ee5c. N\u1ed3ng \u0111\u1ed9 cGMP trong th\u1ec3 hang t\u0103ng do Tadalafil \u1ee9c ch\u1ebf ch\u1ecdn l\u1ecdc PDE5. Do \u0111\u00f3 l\u00e0m gi\u00e3n c\u01a1 tr\u01a1n, t\u0103ng l\u01b0\u1ee3ng m\u00e1u v\u00e0o m\u00f4 d\u01b0\u01a1ng v\u1eadt v\u00e0 l\u00e0m c\u01b0\u01a1ng d\u01b0\u01a1ng v\u1eadt.Tadalafil m\u1ea5t t\u00e1c d\u1ee5ng l\u00e0m c\u01b0\u01a1ng khi kh\u00f4ng c\u00f3 c\u00e1c k\u00edch th\u00edch v\u1ec1 t\u00ecnh d\u1ee5c,.<\/p>\n
\nSo v\u1edbi t\u00e1c d\u1ee5ng tr\u00ean c\u00e1c ch\u1ea5t PDE1, PDE2, PDE3, PDE4 v\u00e0 PDE7 th\u00ec t\u00e1c d\u1ee5ng tr\u00ean PDE5 c\u1ee7a Tadalafil m\u1ea1nh g\u1ea5p >10.000 l\u1ea7n.
\nSo v\u1edbi PDE6, t\u00e1c \u0111\u1ed9ng Tadalafil tr\u00ean PDE5 m\u1ea1nh h\u01a1n kho\u1ea3ng 700 l\u1ea7n, tr\u00ean PDE5 m\u1ea1nh g\u1ea5p >9.000 l\u1ea7n so v\u1edbi PDE 8, PDE9, PDE10.<\/p>\n\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n
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\nTadalafil\u00a0 b\u00e0i ti\u1ebft qua ph\u00e2n kho\u1ea3ng 61% v\u00e0 trong n\u01b0\u1edbc ti\u1ec3u kho\u1ea3ng 36% d\u01b0\u1edbi d\u1ea1ng c\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a kh\u00f4ng c\u00f3 t\u00e1c t\u00e1c d\u1ee5ng.<\/p>\nThu\u1ed1c C.ales 20mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n
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Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c C.ales 20mg<\/h2>\n