{"id":41662,"date":"2023-09-10T23:36:25","date_gmt":"2023-09-10T16:36:25","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=41662"},"modified":"2025-11-03T17:48:52","modified_gmt":"2025-11-03T10:48:52","slug":"thuoc-ckdmyrept-tab-500mg","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/thuoc-ckdmyrept-tab-500mg\/","title":{"rendered":"Ckdmyrept Tab. 500mg"},"content":{"rendered":"
\u00a0Trong b\u00e0i vi\u1ebft n\u00e0y, D\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n th\u00f4ng tin v\u1ec1 thu\u1ed1c Ckdmyrept Tab. 500mg<\/a> ch\u1ee9a ho\u1ea1t ch\u1ea5t Mycophenolate mofetil, \u0111\u01b0\u1ee3c d\u00f9ng d\u1ef1 ph\u00f2ng hi\u1ec7n t\u01b0\u1ee3ng th\u1ea3i gh\u00e9p c\u1ea5p t\u00ednh \u1edf b\u1ec7nh nh\u00e2n v\u1eeba th\u1ef1c hi\u1ec7n gh\u00e9p gan. <\/b>Thu\u1ed1c Ckdmyrept Tab. 500mg \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t v\u00e0 ph\u00e2n ph\u1ed1i b\u1edfi c\u00f4ng ty d\u01b0\u1ee3c ph\u1ea9m Chong Kun Dang Pharmaceutical Corp – H\u00e0n Qu\u1ed1c, hi\u1ec7n \u0111ang c\u00f3 s\u1ed1 l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-17851-14.<\/b><\/p>\n Thu\u1ed1c Ckdmyrept Tab. 500mg <\/b>c\u00f3 ch\u1ee9a th\u00e0nh ph\u1ea7n:<\/span><\/p>\n D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim.<\/p>\n S\u0110K: VN-17851-14.<\/span><\/p>\n Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 10 v\u1ec9 x 10 vi\u00ean.<\/span><\/p>\n Xu\u1ea5t x\u1ee9: H\u00e0n Qu\u1ed1c.<\/span><\/p>\n Mycophenolate mofetil l\u00e0 thu\u1ed1c thu\u1ed9c nh\u00f3m \u1ee9c ch\u1ebf mi\u1ec5n d\u1ecbch,\u00a0c\u00f3 b\u1ea3n ch\u1ea5t l\u00e0 m\u1ed9t ti\u1ec1n ch\u1ea5t c\u1ee7a axit mycophenolic v\u00e0 \u0111\u01b0\u1ee3c ph\u00e2n lo\u1ea1i l\u00e0 ch\u1ea5t \u1ee9c ch\u1ebf c\u00f3 th\u1ec3 \u0111\u1ea3o ng\u01b0\u1ee3c c\u1ee7a Inosine monophosphate\u00a0dehydrogenase (IMPDH).<\/p>\n C\u01a1 ch\u1ebf ho\u1ea1t \u0111\u1ed9ng c\u1ee7a MPA l\u00e0 n\u00f3 \u1ee9c ch\u1ebf enzym Inosine monophosphate Dehydrogenase (IMPDH). \u0110i\u1ec1u n\u00e0y l\u00e0m ng\u0103n c\u1ea3n qu\u00e1 tr\u00ecnh x\u00fac t\u00e1c c\u1ee7a IMPDH \u0111\u1ec3 bi\u1ebfn \u0111\u1ed5i IMP th\u00e0nh xanthose-5\u2019-monophosphate. \u0110\u00e2y \u0111\u01b0\u1ee3c xem nh\u01b0 m\u1ed9t b\u01b0\u1edbc ch\u00ednh trong con \u0111\u01b0\u1eddng denovo c\u1ee7a qu\u00e1 tr\u00ecnh t\u1ed5ng h\u1ee3p Guanosine nucleotide.<\/p>\n T\u00e1c d\u1ee5ng \u1ee9c ch\u1ebf IMPDH l\u00e0 t\u00e1c d\u1ee5ng m\u1ea1nh, ch\u1ecdn l\u1ecdc v\u00e0 c\u00f3 kh\u1ea3 n\u0103ng h\u1ed3i ph\u1ee5c. MPA c\u00f3 t\u00e1c d\u1ee5ng k\u00ecm h\u00e3m m\u1ea1nh c\u00e1c t\u1ebf b\u00e0o lympho B v\u00e0 lympho T h\u01a1n c\u00e1c t\u1ebf b\u00e0o kh\u00e1c do c\u00e1c t\u1ebf b\u00e0o lympho ph\u1ee5 thu\u1ed9c nhi\u1ec1u v\u00e0o con \u0111\u01b0\u1eddng Denovo \u0111\u1ec3 t\u1ed5ng h\u1ee3p Guanosine trong khi c\u00e1c t\u1ebf b\u00e0o kh\u00e1c c\u00f3 th\u1ec3 s\u1eed d\u1ee5ng c\u00e1c con \u0111\u01b0\u1eddng t\u00e1i t\u1ea1o kh\u00e1c.<\/p>\n H\u1ea5p thu: Mycophenolate Mofetil \u0111\u01b0\u1ee3c h\u1ea5p thu nhanh ch\u00f3ng \u1edf ru\u1ed9t non. N\u1ed3ng \u0111\u1ed9 axit mycophenolic \u0111\u1ea1t \u0111\u1ec9nh sau 60 \u0111\u1ebfn 90 ph\u00fat t\u1eeb khi u\u1ed1ng li\u1ec1u \u0111\u1ea7u ti\u00ean. S\u1ef1 h\u1ea5p thu c\u1ee7a thu\u1ed1c kh\u00f4ng b\u1ecb \u1ea3nh h\u01b0\u1edfng b\u1edfi th\u1ee9c \u0103n.<\/p>\n Ph\u00e2n b\u1ed1: Th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 thu\u1ed1c c\u1ee7a Mycophenolate Mofetil l\u00e0 3,6 (\u00b11,5) \u0111\u1ebfn 4,0 (\u00b11,2) L\/kg. T\u1ef7 l\u1ec7 li\u00ean k\u1ebft v\u1edbi protein c\u1ee7a axit mycophenolic, s\u1ea3n ph\u1ea9m chuy\u1ec3n h\u00f3a c\u1ee7a Mycophenolate Mofetil, l\u00e0 97%. Ch\u00fang ch\u1ee7 y\u1ebfu \u0111\u01b0\u1ee3c li\u00ean k\u1ebft v\u1edbi albumin. MPAG, ch\u1ea5t chuy\u1ec3n h\u00f3a kh\u00f4ng c\u00f3 ho\u1ea1t t\u00ednh, li\u00ean k\u1ebft 82% v\u1edbi Albumin huy\u1ebft t\u01b0\u01a1ng \u1edf n\u1ed3ng \u0111\u1ed9 \u0111i\u1ec1u tr\u1ecb th\u00f4ng th\u01b0\u1eddng.<\/p>\n Chuy\u1ec3n h\u00f3a: Sau khi u\u1ed1ng v\u00e0 ti\u00eam t\u0129nh m\u1ea1ch, Mycophenolate Mofetil \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a ho\u00e0n to\u00e0n b\u1edfi carboxylesterase gan 1 v\u00e0 2 th\u00e0nh axit mycophenolic (MPA), c\u00f3 ho\u1ea1t t\u00ednh. Sau \u0111\u00f3, n\u00f3 \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a b\u1edfi enzyme glucuronyl transferase, t\u1ea1o ra phenolic glucuronide kh\u00f4ng ho\u1ea1t \u0111\u1ed9ng c\u1ee7a MPA (MPAG)<\/p>\n Th\u1ea3i tr\u1eeb: M\u1ed9t l\u01b0\u1ee3ng nh\u1ecf thu\u1ed1c \u0111\u01b0\u1ee3c b\u00e0i ti\u1ebft d\u01b0\u1edbi d\u1ea1ng MPA trong n\u01b0\u1edbc ti\u1ec3u (d\u01b0\u1edbi 1%). Kho\u1ea3ng 87% to\u00e0n b\u1ed9 li\u1ec1u d\u00f9ng \u0111\u01b0\u1ee3c b\u00e0i ti\u1ebft qua n\u01b0\u1edbc ti\u1ec3u d\u01b0\u1edbi d\u1ea1ng MPAG, m\u1ed9t ch\u1ea5t chuy\u1ec3n h\u00f3a kh\u00f4ng c\u00f3 ho\u1ea1t t\u00ednh. \u0110\u1ed9 thanh th\u1ea3i huy\u1ebft t\u01b0\u01a1ng c\u1ee7a Mycophenolate Mofetil l\u00e0 193 mL\/ph\u00fat sau li\u1ec1u u\u1ed1ng v\u00e0 177 (\u00b131) mL\/ph\u00fat sau li\u1ec1u ti\u00eam t\u0129nh m\u1ea1ch. N\u1eeda \u0111\u1eddi th\u1ea3i tr\u1eeb bi\u1ec3u ki\u1ebfn \u200b\u200btrung b\u00ecnh c\u1ee7a Mycophenolate Mofetil l\u00e0 17,9 (\u00b16,5) gi\u1edd sau khi u\u1ed1ng v\u00e0 16,6 (\u00b15,8) gi\u1edd sau khi ti\u00eam t\u0129nh m\u1ea1ch.<\/p>\n Thu\u1ed1c\u00a0\u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh s\u1eed d\u1ee5ng k\u1ebft h\u1ee3p v\u1edbi\u00a0Cyclosporine\u00a0va Corticosteroid \u0111\u1ec3 d\u1ef1 ph\u00f2ng hi\u1ec7n t\u01b0\u1ee3ng th\u1ea3i gh\u00e9p c\u1ea5p t\u00ednh, th\u1ea3i gh\u00e9p l\u1ea7n \u0111\u1ea7u, \u0111\u00e1p \u1ee9ng k\u00e9m \u1edf nh\u1eefng b\u1ec7nh nh\u00e2n gh\u00e9p gan kh\u00f4ng c\u00f9ng huy\u1ebft th\u1ed1ng, gh\u00e9p th\u1eadn, gh\u00e9p tim.<\/p>\n Thu\u1ed1c Ckdmyrept Tab. 500mg \u0111\u01b0\u1ee3c b\u00e0o ch\u1ebf d\u01b0\u1edbi d\u1ea1ng vi\u00ean n\u00e9n bao phim do \u0111\u00f3 \u0111\u01b0\u1ee3c d\u00f9ng theo \u0111\u01b0\u1eddng u\u1ed1ng.<\/p>\n N\u00ean u\u1ed1ng thu\u1ed1c v\u1edbi m\u1ed9t c\u1ed1c n\u01b0\u1edbc, tuy\u1ec7t \u0111\u1ed1i kh\u00f4ng \u0111\u01b0\u1ee3c nhai, nghi\u1ec1n.<\/p>\n D\u01b0\u1edbi \u0111\u00e2y l\u00e0 li\u1ec1u l\u01b0\u1ee3ng tham kh\u1ea3o. Li\u1ec1u d\u00f9ng c\u1ee5 th\u1ec3 t\u00f9y thu\u1ed9c v\u00e0o th\u1ec3 tr\u1ea1ng v\u00e0 m\u1ee9c \u0111\u1ed9 di\u1ec5n ti\u1ebfn c\u1ee7a b\u1ec7nh.<\/p>\nCkdmyrept Tab. 500mg l\u00e0 thu\u1ed1c g\u00ec?<\/span><\/h2>\n
Th\u00e0nh ph\u1ea7n<\/span><\/h3>\n
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Tr\u00ecnh b\u00e0y<\/span><\/h3>\n
T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Ckdmyrept Tab. 500mg<\/span><\/h2>\n
D\u01b0\u1ee3c l\u1ef1c h\u1ecdc<\/span><\/h3>\n
D\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc\u00a0<\/span><\/h3>\n
Thu\u1ed1c Ckdmyrept Tab. 500mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/span><\/h2>\n
Li\u1ec1u d\u00f9ng v\u00e0 C\u00e1ch d\u00f9ng c\u1ee7a thu\u1ed1c Ckdmyrept Tab. 500mg<\/span><\/h2>\n
C\u00e1ch d\u00f9ng thu\u1ed1c Ckdmyrept Tab. 500mg<\/h3>\n
Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Ckdmyrept Tab. 500mg<\/h3>\n