{"id":149737,"date":"2025-12-04T13:50:15","date_gmt":"2025-12-04T06:50:15","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=149737"},"modified":"2025-12-04T13:54:31","modified_gmt":"2025-12-04T06:54:31","slug":"ezenstatin-10-10","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/ezenstatin-10-10\/","title":{"rendered":"Ezenstatin 10\/10"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y, <\/strong>d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/strong><\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c Ezenstatin 10\/10<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi<\/strong> Chi nh\u00e1nh c\u00f4ng ty c\u1ed5 ph\u1ea7n d\u01b0\u1ee3c ph\u1ea9m Agimexpharm- Nh\u00e0 m\u00e1y s\u1ea3n xu\u1ea5t d\u01b0\u1ee3c ph\u1ea9m Agimexpharm , c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 893110015500 (S\u0110K c\u0169: VD-32782-19).<\/strong><\/p>\n

Ezenstatin 10\/10 l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

Thu\u1ed1c Ezenstatin 10\/10<\/strong> c\u00f3 ch\u1ee9a th\u00e0nh ph\u1ea7n: Atorvastatin (d\u01b0\u1edbi d\u1ea1ng Atorvastatin calci) 10mg; Ezetimibe 10mg<\/p>\n

D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: 893110015500 (S\u0110K c\u0169: VD-32782-19)<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 4 v\u1ec9 x 7 vi\u00ean<\/p>\n

Xu\u1ea5t x\u1ee9: Vi\u1ec7t Nam<\/p>\n

H\u1ea1n s\u1eed d\u1ee5ng: 36 th\u00e1ng<\/p>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Ezenstatin 10\/10<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

Atorvastatin \u1ee9c ch\u1ebf c\u1ea1nh tranh v\u1edbi HMG CoA, h\u1ea1n ch\u1ebf s\u1ef1 h\u00ecnh th\u00e0nh mevalonat l\u00e0 m\u1ed9t ti\u1ec1n ch\u1ea5t c\u1ee7a cholesterol, \u1ee9c ch\u1ebf qu\u00e1 tr\u00ecnh t\u1ed5ng h\u1ee3p cholesterol, t\u1eeb \u0111\u00f3 gi\u1ea3m l\u01b0\u1ee3ng th\u00e0nh ph\u1ea7n n\u00e0y \u1edf gan. Tuy nhi\u00ean, \u1edf li\u1ec1u \u0111i\u1ec1u tr\u1ecb, Ezetimibe kh\u00f4ng \u1ee9c ch\u1ebf HMG CoA ho\u00e0n to\u00e0n, do \u0111\u00f3 trong c\u01a1 th\u1ec3 v\u1eabn c\u00f3 \u0111\u1ee7 l\u01b0\u1ee3ng acid mevalonic cho c\u00e1c qu\u00e1 tr\u00ecnh chuy\u1ec3n h\u00f3a t\u1ef1 nhi\u00ean.<\/p>\n

Ezetimibe c\u00f3 c\u00f4ng d\u1ee5ng \u1ee9c ch\u1ebf s\u1ef1 h\u1ea5p thu cholesterol \u1edf ru\u1ed9t non, gi\u1ea3m v\u1eadn chuy\u1ec3n cholesterol t\u1eeb ru\u1ed9t v\u00e0o gan, t\u1eeb \u0111\u00f3 h\u1ea1n ch\u1ebf t\u00ecnh tr\u1ea1ng t\u00edch tr\u1eef cholesterol \u1edf gan, t\u0103ng c\u01b0\u1eddng th\u1ea3i cholesterol kh\u1ecfi m\u00e1u, t\u1eeb \u0111\u00f3 h\u1ed7 tr\u1ee3 n\u00e2ng cao c\u00f4ng d\u1ee5ng c\u1ee7a ho\u1ea1t ch\u1ea5t nh\u00f3n statin.<\/p>\n

\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

Atorvastatin h\u1ea5p thu nhanh ch\u00f3ng khi d\u00f9ng \u0111\u01b0\u1eddng u\u1ed1ng v\u00e0 kh\u00f4ng b\u1ecb t\u00e1c \u0111\u1ed9ng b\u1edfi s\u1ef1 c\u00f3 m\u1eb7t c\u1ee7a th\u1ee9c \u0103n, n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh c\u1ee7a thu\u1ed1c \u0111\u01b0\u1ee3c ghi nh\u1eadn sau 1-2 gi\u1edd. Sinh kh\u1ea3 d\u1ee5ng tuy\u1ec7t \u0111\u1ed1i th\u1ea5p, ch\u1ec9 kho\u1ea3ng 14%. Kho\u1ea3ng 98% Atorvastatin li\u00ean k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng. Sau khi v\u00e0o c\u01a1 th\u1ec3, ho\u1ea1t ch\u1ea5t \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a ch\u00ednh gan, tr\u00ean 70% li\u1ec1u d\u00f9ng, t\u1ea1o th\u00e0nh c\u00e1c ch\u1ea5t c\u00f3 ho\u1eb7c kh\u00f4ng c\u00f3 ho\u1ea1t t\u00ednh, sau \u0111\u00f3 th\u1ea3i tr\u1eeb qua ph\u00e2n.<\/p>\n

Ezetimibe h\u1ea5p thu nhanh ch\u00f3ng khi d\u00f9ng \u0111\u01b0\u1eddng u\u1ed1ng v\u00e0 t\u1ea1o th\u00e0nh d\u1ea1ng li\u00ean h\u1ee3p Ezetimibe glucuronid. Ho\u1ea1t ch\u1ea5t g\u1ed1c chuy\u1ec3n h\u00f3a ch\u1ee7 y\u1ebfu \u1edf ru\u1ed9t non v\u00e0 gan, sau \u0111\u00f3 th\u1ea3i tr\u1eeb qua ph\u00e2n v\u00e0 n\u01b0\u1edbc ti\u1ec3u.<\/p>\n\n\n\n\n\n\n
<\/td>\nEzetimibe<\/td>\nEzetimibe glucuronid<\/td>\n<\/tr>\n
Th\u1eddi gian \u0111\u1ea1t n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng<\/td>\n1-2 gi\u1edd<\/td>\n4-12 gi\u1edd<\/td>\n<\/tr>\n
T\u1ef7 l\u1ec7 li\u00ean k\u1ebft protein huy\u1ebft t\u01b0\u01a1ng<\/td>\n99,7%<\/td>\n88-92%<\/td>\n<\/tr>\n
Th\u1eddi gian b\u00e1n th\u1ea3i<\/td>\n22 gi\u1edd<\/td>\n22 gi\u1edd<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n

Thu\u1ed1c Ezenstatin 10\/10 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

Thu\u1ed1c Ezenstatin 10\/10<\/strong> d\u00f9ng trong d\u1ef1 ph\u00f2ng bi\u1ebfn c\u1ed1 tim m\u1ea1ch \u1edf b\u1ec7nh nh\u00e2n b\u1ecb b\u1ec7nh m\u1ea1ch v\u00e0nh v\u00e0 \u0111i\u1ec1u tr\u1ecb t\u0103ng cholesterol m\u00e1u (bao g\u1ed3m c\u1ea3 t\u0103ng cholesterol m\u00e1u nguy\u00ean ph\u00e1t v\u00e0 t\u0103ng cholesterol m\u00e1u gia \u0111\u00ecnh ki\u1ec3u \u0111\u1ed3ng h\u1ee3p t\u1eed)<\/p>\n

\"Thu\u1ed1c
Thu\u1ed1c Ezenstatin 10\/10 \u2013 \u0110i\u1ec1u tr\u1ecb t\u0103ng cholesterol m\u00e1u nguy\u00ean ph\u00e1t<\/figcaption><\/figure>\n

Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Ezenstatin 10\/10<\/h2>\n

Li\u1ec1u d\u00f9ng<\/h3>\n