{"id":139218,"date":"2025-09-16T12:47:58","date_gmt":"2025-09-16T05:47:58","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=139218"},"modified":"2025-09-16T12:49:06","modified_gmt":"2025-09-16T05:49:06","slug":"omeptul-20mg","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/omeptul-20mg\/","title":{"rendered":"Omeptul 20mg"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y,<\/strong> d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/strong><\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c<\/strong> Omeptul 20mg<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi Gracure Pharmaceuticals Ltd., c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-12327-11.<\/strong><\/p>\n

Omeptul 20mg l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

Omeptul 20mg<\/strong> l\u00e0 m\u1ed9t thu\u1ed1c thu\u1ed9c nh\u00f3m \u1ee9c ch\u1ebf b\u01a1m proton (Proton Pump Inhibitor – PPI), m\u1ed7i vi\u00ean nang ch\u1ee9a Omeprazole <\/strong>20mg (d\u01b0\u1edbi d\u1ea1ng c\u00e1c vi h\u1ea1t bao tan trong ru\u1ed9t).<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: VN-12327-11<\/p>\n

D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean nang<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 10 v\u1ec9 x 10 vi\u00ean<\/p>\n

Xu\u1ea5t x\u1ee9: \u1ea4n \u0110\u1ed9<\/p>\n

\"Omeptul
Omeptul 20mg \u0111i\u1ec1u tr\u1ecb tr\u00e0o ng\u01b0\u1ee3c d\u1ecbch d\u1ea1 d\u00e0y – th\u1ef1c qu\u1ea3n<\/figcaption><\/figure>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Omeptul 20mg<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

Omeprazole l\u00e0 m\u1ed9t ti\u1ec1n ch\u1ea5t (prodrug), sau khi \u0111\u01b0\u1ee3c h\u1ea5p thu v\u00e0o m\u00e1u s\u1ebd t\u1eadp trung t\u1ea1i c\u00e1c t\u1ebf b\u00e0o th\u00e0nh c\u1ee7a d\u1ea1 d\u00e0y (parietal cells) \u2013 n\u01a1i s\u1ea3n xu\u1ea5t acid. Trong m\u00f4i tr\u01b0\u1eddng acid cao \u0111\u1ed9 c\u1ee7a t\u1ebf b\u00e0o th\u00e0nh, Omeprazole \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a th\u00e0nh d\u1ea1ng ho\u1ea1t \u0111\u1ed9ng l\u00e0 sulfenamide. Ch\u1ea5t n\u00e0y sau \u0111\u00f3 li\u00ean k\u1ebft kh\u00f4ng thu\u1eadn ngh\u1ecbch v\u1edbi nh\u00f3m sulfhydryl (-SH) c\u1ee7a enzym H+\/K+-ATPase, hay c\u00f2n g\u1ecdi l\u00e0 b\u01a1m proton.<\/p>\n

Enzym n\u00e0y l\u00e0 kh\u00e2u cu\u1ed1i c\u00f9ng v\u00e0 quan tr\u1ecdng nh\u1ea5t trong qu\u00e1 tr\u00ecnh b\u00e0i ti\u1ebft acid hydrochloric (HCl) v\u00e0o l\u00f2ng d\u1ea1 d\u00e0y. B\u1eb1ng c\u00e1ch \u1ee9c ch\u1ebf v\u0129nh vi\u1ec5n b\u01a1m proton, Omeprazole ng\u0103n ch\u1eb7n hi\u1ec7u qu\u1ea3 c\u1ea3 s\u1ef1 ti\u1ebft acid c\u01a1 b\u1ea3n (l\u00fac \u0111\u00f3i) v\u00e0 khi \u0111\u01b0\u1ee3c k\u00edch th\u00edch (b\u1edfi th\u1ee9c \u0103n, histamine, gastrin). T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c k\u00e9o d\u00e0i cho \u0111\u1ebfn khi c\u00e1c b\u01a1m proton m\u1edbi \u0111\u01b0\u1ee3c t\u1ed5ng h\u1ee3p, th\u01b0\u1eddng l\u00e0 sau 24 gi\u1edd, gi\u00fap ki\u1ec3m so\u00e1t acid d\u1ea1 d\u00e0y su\u1ed1t c\u1ea3 ng\u00e0y ch\u1ec9 v\u1edbi m\u1ed9t li\u1ec1u duy nh\u1ea5t.<\/p>\n

\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

H\u1ea5p thu: Omeprazole kh\u00f4ng b\u1ec1n trong m\u00f4i tr\u01b0\u1eddng acid, do \u0111\u00f3 thu\u1ed1c \u0111\u01b0\u1ee3c b\u00e0o ch\u1ebf d\u01b0\u1edbi d\u1ea1ng vi h\u1ea1t bao tan trong ru\u1ed9t \u0111\u1ec3 b\u1ea3o v\u1ec7 ho\u1ea1t ch\u1ea5t kh\u1ecfi s\u1ef1 ph\u00e1 h\u1ee7y c\u1ee7a d\u1ecbch v\u1ecb v\u00e0 ch\u1ec9 tan ra \u1edf m\u00f4i tr\u01b0\u1eddng ki\u1ec1m c\u1ee7a ru\u1ed9t non. Thu\u1ed1c \u0111\u01b0\u1ee3c h\u1ea5p thu nhanh, n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng \u0111\u1ea1t \u0111\u01b0\u1ee3c sau 1-2 gi\u1edd.<\/p>\n

Ph\u00e2n b\u1ed1: Kho\u1ea3ng 97% Omeprazole li\u00ean k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng.<\/p>\n

Chuy\u1ec3n h\u00f3a: Thu\u1ed1c \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a g\u1ea7n nh\u01b0 ho\u00e0n to\u00e0n t\u1ea1i gan, ch\u1ee7 y\u1ebfu qua h\u1ec7 th\u1ed1ng enzyme cytochrome P450, c\u1ee5 th\u1ec3 l\u00e0 isoenzyme CYP2C19 v\u00e0 CYP3A4.<\/p>\n

Th\u1ea3i tr\u1eeb: C\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb ch\u1ee7 y\u1ebfu qua n\u01b0\u1edbc ti\u1ec3u (kho\u1ea3ng 80%) v\u00e0 m\u1ed9t ph\u1ea7n qua ph\u00e2n. M\u1eb7c d\u00f9 th\u1eddi gian b\u00e1n th\u1ea3i trong huy\u1ebft t\u01b0\u01a1ng ng\u1eafn (kho\u1ea3ng 1-2 gi\u1edd), t\u00e1c d\u1ee5ng \u1ee9c ch\u1ebf ti\u1ebft acid l\u1ea1i k\u00e9o d\u00e0i do s\u1ef1 li\u00ean k\u1ebft kh\u00f4ng thu\u1eadn ngh\u1ecbch v\u1edbi b\u01a1m proton.<\/p>\n

Thu\u1ed1c Omeptul 20mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

B\u1ec7nh tr\u00e0o ng\u01b0\u1ee3c d\u1ea1 d\u00e0y-th\u1ef1c qu\u1ea3n (GERD): \u0110i\u1ec1u tr\u1ecb vi\u00eam th\u1ef1c qu\u1ea3n do tr\u00e0o ng\u01b0\u1ee3c v\u00e0 ki\u1ec3m so\u00e1t c\u00e1c tri\u1ec7u ch\u1ee9ng nh\u01b0 \u1ee3 n\u00f3ng, \u1ee3 chua.<\/p>\n

Lo\u00e9t d\u1ea1 d\u00e0y-t\u00e1 tr\u00e0ng: \u0110i\u1ec1u tr\u1ecb v\u00e0 ph\u00f2ng ng\u1eeba t\u00e1i ph\u00e1t lo\u00e9t d\u1ea1 d\u00e0y, lo\u00e9t t\u00e1 tr\u00e0ng.<\/p>\n

Ph\u1ed1i h\u1ee3p di\u1ec7t tr\u1eeb vi khu\u1ea9n Helicobacter pylori<\/em> (H. pylori): L\u00e0 m\u1ed9t th\u00e0nh ph\u1ea7n quan tr\u1ecdng trong c\u00e1c ph\u00e1c \u0111\u1ed3 \u0111a kh\u00e1ng sinh \u0111\u1ec3 ti\u1ec7t tr\u1eeb H. pylori<\/em>, nguy\u00ean nh\u00e2n ch\u00ednh g\u00e2y lo\u00e9t d\u1ea1 d\u00e0y-t\u00e1 tr\u00e0ng.<\/p>\n

H\u1ed9i ch\u1ee9ng Zollinger-Ellison: \u0110i\u1ec1u tr\u1ecb t\u00ecnh tr\u1ea1ng t\u0103ng ti\u1ebft acid b\u1ec7nh l\u00fd hi\u1ebfm g\u1eb7p do kh\u1ed1i u gastrinoma.<\/p>\n

Ph\u00f2ng v\u00e0 \u0111i\u1ec1u tr\u1ecb lo\u00e9t do thu\u1ed1c kh\u00e1ng vi\u00eam kh\u00f4ng steroid (NSAIDs): D\u00e0nh cho nh\u1eefng b\u1ec7nh nh\u00e2n c\u00f3 nguy c\u01a1 cao c\u1ea7n s\u1eed d\u1ee5ng NSAIDs k\u00e9o d\u00e0i.<\/p>\n

Li\u1ec1u d\u00f9ng v\u00e0 c\u00e1ch d\u00f9ng c\u1ee7a thu\u1ed1c Omeptul 20mg<\/h2>\n

Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Omeptul 20mg<\/h3>\n

Li\u1ec1u d\u00f9ng d\u01b0\u1edbi \u0111\u00e2y ch\u1ec9 mang t\u00ednh tham kh\u1ea3o v\u00e0 c\u1ea7n \u0111\u01b0\u1ee3c c\u00e1 nh\u00e2n h\u00f3a theo ch\u1ec9 \u0111\u1ecbnh c\u1ee7a b\u00e1c s\u0129.<\/p>\n