{"id":134186,"date":"2025-08-22T10:02:24","date_gmt":"2025-08-22T03:02:24","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=134186"},"modified":"2026-01-04T12:55:49","modified_gmt":"2026-01-04T05:55:49","slug":"mydocalm-50mg","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/mydocalm-50mg\/","title":{"rendered":"Mydocalm 50mg"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y,<\/strong> d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/strong><\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c<\/strong> Mydocalm 50mg \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi Gedeon Richter Plc., c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-19158-15.<\/strong><\/p>\n

Mydocalm 50mg l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

Mydocalm 50mg <\/strong>l\u00e0 m\u1ed9t thu\u1ed1c gi\u00e3n c\u01a1 t\u00e1c d\u1ee5ng trung \u01b0\u01a1ng, c\u00f3 th\u00e0nh ph\u1ea7n bao g\u1ed3m:<\/p>\n\n\n\n\n
Ho\u1ea1t ch\u1ea5t<\/td>\nTolperisone<\/strong> hydrochloride 50mg<\/td>\n<\/tr>\n
T\u00e1 d\u01b0\u1ee3c<\/td>\nL\u00f5i vi\u00ean: Acid citric monohydrat, silica khan d\u1ea1ng keo, acid stearic, talc, cellulose vi tinh th\u1ec3, tinh b\u1ed9t ng\u00f4, lactose monohydrat.<\/p>\n

L\u1edbp bao: Silica khan d\u1ea1ng keo, titan dioxid (E171), macrogol 600, hypromellose, lactose monohydrat.<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: VN-19158-15<\/p>\n

D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 3 v\u1ec9 x 10 vi\u00ean n\u00e9n bao phim<\/p>\n

Xu\u1ea5t x\u1ee9: Hungary<\/p>\n

\"Mydocalm
Mydocalm 50mg \u0111i\u1ec1u tr\u1ecb tri\u1ec7u ch\u1ee9ng co c\u1ee9ng c\u01a1 sau \u0111\u1ed9t qu\u1ef5<\/figcaption><\/figure>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Mydocalm 50mg<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng ch\u00ednh x\u00e1c c\u1ee7a Tolperisone v\u1eabn \u0111ang \u0111\u01b0\u1ee3c nghi\u00ean c\u1ee9u, tuy nhi\u00ean c\u00e1c b\u1eb1ng ch\u1ee9ng khoa h\u1ecdc cho th\u1ea5y thu\u1ed1c t\u00e1c \u0111\u1ed9ng th\u00f4ng qua m\u1ed9t c\u01a1 ch\u1ebf ph\u1ee9c h\u1ee3p v\u00e0 \u0111a \u0111i\u1ec3m:<\/p>\n

    \n
  • \u1ed4n \u0111\u1ecbnh m\u00e0ng t\u1ebf b\u00e0o th\u1ea7n kinh: Tolperisone c\u00f3 t\u00e1c d\u1ee5ng g\u00e2y t\u00ea c\u1ee5c b\u1ed9, gi\u00fap \u1ed5n \u0111\u1ecbnh m\u00e0ng t\u1ebf b\u00e0o c\u1ee7a c\u00e1c s\u1ee3i th\u1ea7n kinh c\u1ea3m gi\u00e1c nguy\u00ean ph\u00e1t v\u00e0 c\u00e1c n\u01a1ron v\u1eadn \u0111\u1ed9ng. T\u00e1c \u0111\u1ed9ng n\u00e0y \u0111\u01b0\u1ee3c th\u1ef1c hi\u1ec7n th\u00f4ng qua vi\u1ec7c \u1ee9c ch\u1ebf c\u00e1c k\u00eanh ion natri (Na+) v\u00e0 calci (Ca2+) ph\u1ee5 thu\u1ed9c \u0111i\u1ec7n th\u1ebf. B\u1eb1ng c\u00e1ch ch\u1eb9n c\u00e1c k\u00eanh n\u00e0y, Tolperisone l\u00e0m gi\u1ea3m s\u1ef1 kh\u1eed c\u1ef1c c\u1ee7a m\u00e0ng t\u1ebf b\u00e0o, t\u1eeb \u0111\u00f3 ng\u0103n ch\u1eb7n s\u1ef1 h\u00ecnh th\u00e0nh v\u00e0 lan truy\u1ec1n c\u1ee7a c\u00e1c \u0111i\u1ec7n th\u1ebf ho\u1ea1t \u0111\u1ed9ng, l\u00e0m \u1ee9c ch\u1ebf s\u1ef1 d\u1eabn truy\u1ec1n t\u00edn hi\u1ec7u th\u1ea7n kinh g\u00e2y co c\u01a1.<\/li>\n
  • \u1ee8c ch\u1ebf ph\u1ea3n x\u1ea1 t\u1ee7y s\u1ed1ng: T\u1ea1i t\u1ee7y s\u1ed1ng, vi\u1ec7c \u1ee9c ch\u1ebf d\u00f2ng Ca2+ v\u00e0o \u0111\u1ea7u t\u1eadn c\u00f9ng synap s\u1ebd ng\u0103n c\u1ea3n s\u1ef1 gi\u1ea3i ph\u00f3ng c\u00e1c ch\u1ea5t d\u1eabn truy\u1ec1n th\u1ea7n kinh. \u0110i\u1ec1u n\u00e0y d\u1eabn \u0111\u1ebfn \u1ee9c ch\u1ebf hi\u1ec7u qu\u1ea3 c\u1ea3 c\u00e1c cung ph\u1ea3n x\u1ea1 \u0111\u01a1n synap v\u00e0 \u0111a synap, l\u00e0 c\u01a1 s\u1edf cho t\u00e1c d\u1ee5ng gi\u00e3n c\u01a1 c\u1ee7a thu\u1ed1c.<\/li>\n
  • T\u00e1c \u0111\u1ed9ng tr\u00ean th\u00e2n n\u00e3o: Tolperisone c\u00f2n c\u00f3 kh\u1ea3 n\u0103ng \u1ee9c ch\u1ebf \u0111\u01b0\u1eddng ph\u1ea3n x\u1ea1 l\u01b0\u1edbi – t\u1ee7y s\u1ed1ng (reticulospinal tract) \u1edf th\u00e2n n\u00e3o, g\u00f3p ph\u1ea7n l\u00e0m gi\u1ea3m tr\u01b0\u01a1ng l\u1ef1c c\u01a1 qu\u00e1 m\u1ee9c.<\/li>\n<\/ul>\n

    M\u1ed9t \u0111\u1eb7c t\u00ednh d\u01b0\u1ee3c l\u00fd quan tr\u1ecdng c\u1ee7a Tolperisone l\u00e0 thu\u1ed1c c\u00f3 \u00e1i l\u1ef1c th\u1ea5p v\u1edbi h\u1ec7 th\u1ed1ng l\u01b0\u1edbi ho\u1ea1t h\u00f3a (reticular activating system). Do \u0111\u00f3, thu\u1ed1c c\u00f3 t\u00e1c d\u1ee5ng an th\u1ea7n kh\u00f4ng \u0111\u00e1ng k\u1ec3, m\u1ed9t \u01b0u \u0111i\u1ec3m v\u01b0\u1ee3t tr\u1ed9i so v\u1edbi c\u00e1c thu\u1ed1c gi\u00e3n c\u01a1 trung \u01b0\u01a1ng kh\u00e1c nh\u01b0 Baclofen hay Tizanidine, gi\u00fap b\u1ec7nh nh\u00e2n tr\u00e1nh \u0111\u01b0\u1ee3c t\u00ecnh tr\u1ea1ng bu\u1ed3n ng\u1ee7 v\u00e0 m\u1ec7t m\u1ecfi.<\/p>\n

    \u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

    H\u1ea5p thu: Tolperisone \u0111\u01b0\u1ee3c h\u1ea5p thu t\u1ed1t qua ru\u1ed9t non, tuy nhi\u00ean, do b\u1ecb chuy\u1ec3n h\u00f3a l\u1ea7n \u0111\u1ea7u qua gan r\u1ea5t m\u1ea1nh, sinh kh\u1ea3 d\u1ee5ng \u0111\u01b0\u1eddng u\u1ed1ng ch\u1ec9 \u0111\u1ea1t kho\u1ea3ng 20%.<\/p>\n

    \u1ea2nh h\u01b0\u1edfng c\u1ee7a th\u1ee9c \u0103n: Sinh kh\u1ea3 d\u1ee5ng c\u1ee7a Tolperisone t\u0103ng l\u00ean \u0111\u00e1ng k\u1ec3 khi d\u00f9ng c\u00f9ng b\u1eefa \u0103n. M\u1ed9t b\u1eefa \u0103n gi\u00e0u ch\u1ea5t b\u00e9o c\u00f3 th\u1ec3 l\u00e0m t\u0103ng sinh kh\u1ea3 d\u1ee5ng l\u00ean \u0111\u1ebfn 100% v\u00e0 t\u0103ng n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng (Cmax) kho\u1ea3ng 45% so v\u1edbi khi d\u00f9ng thu\u1ed1c l\u00fac \u0111\u00f3i.<\/p>\n

    Chuy\u1ec3n h\u00f3a: Thu\u1ed1c \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a m\u1ea1nh m\u1ebd t\u1ea1i gan, ch\u1ee7 y\u1ebfu qua isoenzyme CYP2D6 c\u1ee7a h\u1ec7 th\u1ed1ng Cytochrome P450, v\u00e0 m\u1ed9t ph\u1ea7n nh\u1ecf qua CYP2C19 v\u00e0 CYP1A2.<\/p>\n

    Th\u1ea3i tr\u1eeb: H\u01a1n 99% li\u1ec1u d\u00f9ng \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb qua th\u1eadn d\u01b0\u1edbi d\u1ea1ng c\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a kh\u00f4ng c\u00f2n ho\u1ea1t t\u00ednh.<\/p>\n

    Thu\u1ed1c Mydocalm 50mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

    Theo gi\u1ea5y ph\u00e9p l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam, Mydocalm 50mg \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh cho:<\/p>\n