{"id":130762,"date":"2025-08-05T11:31:08","date_gmt":"2025-08-05T04:31:08","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=130762"},"modified":"2025-08-05T16:11:55","modified_gmt":"2025-08-05T09:11:55","slug":"xelostad-20","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/xelostad-20\/","title":{"rendered":"Xelostad 20"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y,<\/strong> d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/strong><\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c<\/strong> Xelostad 20 \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi C\u00f4ng ty TNHH Li\u00ean Doanh Stellapharm – chi nh\u00e1nh 1, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VD-35501-21.<\/strong><\/p>\n

Xelostad 20 l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

Trong vi\u00ean n\u00e9n bao phim Xelostad 20<\/strong> c\u00f3 ch\u1ee9a ho\u1ea1t ch\u1ea5t ch\u00ednh Rivaroxaban<\/strong> 20mg v\u00e0 t\u00e1 d\u01b0\u1ee3c v\u1eeba \u0111\u1ee7 1 vi\u00ean.<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: VD-35501-21<\/p>\n

D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 1 v\u1ec9 x 14 vi\u00ean; H\u1ed9p 3 v\u1ec9 x 14 vi\u00ean; H\u1ed9p 8 v\u1ec9 x 14 vi\u00ean.<\/p>\n

Xu\u1ea5t x\u1ee9: Vi\u1ec7t Nam<\/p>\n

\"Xelostad
Xelostad 20 d\u1ef1 ph\u00f2ng \u0111\u1ed9t qu\u1ef5 v\u00e0 thuy\u00ean t\u1eafc m\u1ea1ch to\u00e0n th\u00e2n<\/figcaption><\/figure>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Xelostad 20<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

\u0110\u1ec3 hi\u1ec3u t\u00e1c d\u1ee5ng c\u1ee7a Xelostad 20, c\u1ea7n n\u1eafm r\u00f5 v\u1ec1 con \u0111\u01b0\u1eddng \u0111\u00f4ng m\u00e1u. Qu\u00e1 tr\u00ecnh n\u00e0y l\u00e0 m\u1ed9t chu\u1ed7i ph\u1ea3n \u1ee9ng ph\u1ee9c t\u1ea1p, gi\u1ed1ng nh\u01b0 m\u1ed9t d\u00f2ng th\u00e1c, v\u1edbi s\u1ef1 tham gia c\u1ee7a nhi\u1ec1u y\u1ebfu t\u1ed1. Y\u1ebfu t\u1ed1 Xa (Factor Xa) \u0111\u00f3ng vai tr\u00f2 l\u00e0 m\u1ed9t \u0111i\u1ec3m h\u1ed9i t\u1ee5 then ch\u1ed1t, n\u01a1i c\u1ea3 hai con \u0111\u01b0\u1eddng \u0111\u00f4ng m\u00e1u n\u1ed9i sinh v\u00e0 ngo\u1ea1i sinh g\u1eb7p nhau. Khi \u0111\u01b0\u1ee3c ho\u1ea1t h\u00f3a, Y\u1ebfu t\u1ed1 Xa s\u1ebd chuy\u1ec3n Prothrombin th\u00e0nh Thrombin \u2013 enzyme trung t\u00e2m c\u00f3 kh\u1ea3 n\u0103ng chuy\u1ec3n Fibrinogen (d\u1ea1ng h\u00f2a tan) th\u00e0nh Fibrin (d\u1ea1ng s\u1ee3i kh\u00f4ng tan), t\u1ea1o th\u00e0nh m\u1ea1ng l\u01b0\u1edbi b\u1eaft gi\u1eef c\u00e1c t\u1ebf b\u00e0o m\u00e1u \u0111\u1ec3 h\u00ecnh th\u00e0nh c\u1ee5c m\u00e1u \u0111\u00f4ng (huy\u1ebft kh\u1ed1i).<\/p>\n

Rivaroxaban trong Xelostad 20 ho\u1ea1t \u0111\u1ed9ng b\u1eb1ng c\u00e1ch \u1ee9c ch\u1ebf tr\u1ef1c ti\u1ebfp, ch\u1ecdn l\u1ecdc v\u00e0 c\u00f3 h\u1ed3i ph\u1ee5c ngay t\u1ea1i v\u1ecb tr\u00ed ho\u1ea1t \u0111\u1ed9ng c\u1ee7a Y\u1ebfu t\u1ed1 Xa. B\u1eb1ng c\u00e1ch “kh\u00f3a” Y\u1ebfu t\u1ed1 Xa, Rivaroxaban ng\u0103n ch\u1eb7n hi\u1ec7u qu\u1ea3 qu\u00e1 tr\u00ecnh s\u1ea3n sinh Thrombin, t\u1eeb \u0111\u00f3 l\u00e0m gi\u00e1n \u0111o\u1ea1n s\u1ef1 h\u00ecnh th\u00e0nh v\u00e0 ph\u00e1t tri\u1ec3n c\u1ee7a c\u1ee5c m\u00e1u \u0111\u00f4ng. \u0110\u00e2y l\u00e0 m\u1ed9t c\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng ti\u00ean ti\u1ebfn, c\u00f3 t\u00ednh d\u1ef1 \u0111o\u00e1n cao v\u00e0 kh\u00f4ng c\u1ea7n theo d\u00f5i x\u00e9t nghi\u1ec7m \u0111\u00f4ng m\u00e1u th\u01b0\u1eddng quy nh\u01b0 c\u00e1c thu\u1ed1c kh\u00e1ng Vitamin K truy\u1ec1n th\u1ed1ng.<\/p>\n

\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

H\u1ea5p thu: Rivaroxaban \u0111\u01b0\u1ee3c h\u1ea5p thu nhanh ch\u00f3ng sau khi u\u1ed1ng. \u0110\u1ed1i v\u1edbi li\u1ec1u 20mg, sinh kh\u1ea3 d\u1ee5ng \u0111\u01b0\u1eddng u\u1ed1ng r\u1ea5t cao (80-100%) khi \u0111\u01b0\u1ee3c d\u00f9ng chung v\u1edbi b\u1eefa \u0103n. Th\u1ee9c \u0103n gi\u00fap t\u0103ng kh\u1ea3 n\u0103ng h\u1ea5p thu c\u1ee7a thu\u1ed1c m\u1ed9t c\u00e1ch \u0111\u00e1ng k\u1ec3.<\/p>\n

Ph\u00e2n b\u1ed1: Thu\u1ed1c li\u00ean k\u1ebft m\u1ea1nh v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng (kho\u1ea3ng 92-95%), ch\u1ee7 y\u1ebfu l\u00e0 albumin.<\/p>\n

Chuy\u1ec3n h\u00f3a: Kho\u1ea3ng 2\/3 li\u1ec1u Rivaroxaban \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a qua gan, ch\u1ee7 y\u1ebfu th\u00f4ng qua h\u1ec7 enzyme Cytochrome P450 (CYP3A4, CYP2J2).<\/p>\n

Th\u1ea3i tr\u1eeb: Thu\u1ed1c \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb qua hai con \u0111\u01b0\u1eddng ch\u00ednh: kho\u1ea3ng 1\/3 li\u1ec1u \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb tr\u1ef1c ti\u1ebfp qua th\u1eadn d\u01b0\u1edbi d\u1ea1ng kh\u00f4ng \u0111\u1ed5i v\u00e0 2\/3 c\u00f2n l\u1ea1i \u0111\u01b0\u1ee3c th\u1ea3i tr\u1eeb d\u01b0\u1edbi d\u1ea1ng ch\u1ea5t chuy\u1ec3n h\u00f3a (m\u1ed9t n\u1eeda qua th\u1eadn, m\u1ed9t n\u1eeda qua ph\u00e2n). Th\u1eddi gian b\u00e1n th\u1ea3i c\u1ee7a thu\u1ed1c \u1edf ng\u01b0\u1eddi tr\u1ebb l\u00e0 5-9 gi\u1edd v\u00e0 \u1edf ng\u01b0\u1eddi cao tu\u1ed5i l\u00e0 11-13 gi\u1edd.<\/p>\n

Thu\u1ed1c Xelostad 20 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

Xelostad 20 \u0111\u01b0\u1ee3c c\u1ea5p ph\u00e9p cho c\u00e1c ch\u1ec9 \u0111\u1ecbnh ch\u00ednh sau \u0111\u00e2y \u1edf ng\u01b0\u1eddi tr\u01b0\u1edfng th\u00e0nh:<\/p>\n