{"id":127226,"date":"2025-07-15T16:27:45","date_gmt":"2025-07-15T09:27:45","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=127226"},"modified":"2025-07-28T12:24:27","modified_gmt":"2025-07-28T05:24:27","slug":"atirin-suspension","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/atirin-suspension\/","title":{"rendered":"Atirin Suspension"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y, d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n thu\u1ed1c Atirin Suspension \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi C\u00f4ng ty C\u1ed5 ph\u1ea7n D\u01b0\u1ee3c ph\u1ea9m An Thi\u00ean, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 893110288400 (S\u0110K c\u0169: VD-34136-20)<\/strong><\/p>\n

Atirin Suspension l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

Ebastin 1mg\/ml (0,1% (w\/v))<\/p>\n

T\u00e1 d\u01b0\u1ee3c v\u1eeba \u0111\u1ee7<\/p>\n

D\u1ea1ng b\u00e0o ch\u1ebf: H\u1ed7n d\u1ecbch u\u1ed1ng<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: 893110288400 (S\u0110K c\u0169: VD-34136-20)<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 30 \u1ed1ng x 5ml<\/p>\n

Xu\u1ea5t x\u1ee9: Vi\u1ec7t Nam<\/p>\n

\"Thu\u1ed1c
Thu\u1ed1c Atirin Suspension c\u00f3 t\u00e1c d\u1ee5ng gi\u00fap \u0111i\u1ec1u tr\u1ecb vi\u00eam m\u0169i d\u1ecb \u1ee9ng, c\u00f3 ho\u1eb7c kh\u00f4ng k\u00e8m vi\u00eam k\u1ebft m\u1ea1c<\/figcaption><\/figure>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Atirin Suspension<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

Ebastin l\u00e0 thu\u1ed1c kh\u00e1ng histamin H1 th\u1ebf h\u1ec7 m\u1edbi, c\u00f3 t\u00e1c d\u1ee5ng ch\u1ecdn l\u1ecdc, kh\u1edfi ph\u00e1t nhanh v\u00e0 k\u00e9o d\u00e0i. Ebastin v\u00e0 c\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a c\u1ee7a n\u00f3 kh\u00f4ng qua h\u00e0ng r\u00e0o m\u00e1u n\u00e3o, do \u0111\u00f3 kh\u00f4ng \u1ea3nh h\u01b0\u1edfng l\u00ean th\u1ea7n kinh trung \u01b0\u01a1ng. Hi\u1ec7u l\u1ef1c kh\u00e1ng histamin xu\u1ea5t hi\u1ec7n sau khi u\u1ed1ng v\u00e0 k\u00e9o d\u00e0i kho\u1ea3ng 48 gi\u1edd. Sau khi d\u00f9ng li\u00ean t\u1ee5c 5 ng\u00e0y, t\u00e1c d\u1ee5ng v\u1eabn c\u00f2n trong v\u00f2ng 72 gi\u1edd sau khi ng\u01b0ng thu\u1ed1c, hi\u1ec7u qu\u1ea3 kh\u00f4ng thay \u0111\u1ed5i khi d\u00f9ng k\u00e9o d\u00e0i. Li\u1ec1u t\u1eeb 10 mg m\u1ed7i ng\u00e0y cho th\u1ea5y hi\u1ec7u qu\u1ea3 r\u00f5 r\u1ec7t, t\u00e1c d\u1ee5ng nhanh v\u00e0 b\u1ec1n v\u1eefng. \u1ede li\u1ec1u \u0111i\u1ec1u tr\u1ecb, ebastin kh\u00f4ng k\u00e9o d\u00e0i kho\u1ea3ng QT tuy nhi\u00ean, li\u1ec1u cao nh\u01b0 100 mg\/ng\u00e0y ho\u1eb7c 500 mg li\u1ec1u \u0111\u01a1n c\u00f3 th\u1ec3 l\u00e0m tim \u0111\u1eadp nhanh nh\u1eb9 v\u00e0 r\u00fat ng\u1eafn kho\u1ea3ng QT, nh\u01b0ng kh\u00f4ng \u1ea3nh h\u01b0\u1edfng \u0111\u1ebfn QTc.<\/p>\n

\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

H\u1ea5p thu: Ebastin h\u1ea5p thu nhanh qua \u0111\u01b0\u1eddng ti\u00eau h\u00f3a; d\u00f9ng k\u00e8m b\u1eefa \u0103n gi\u00e0u ch\u1ea5t b\u00e9o l\u00e0m t\u0103ng h\u1ea5p thu v\u00e0 t\u0103ng g\u1eafn k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng kho\u1ea3ng 50%.<\/p>\n

Ph\u00e2n b\u1ed1: Sau li\u1ec1u u\u1ed1ng Ebastin 10mg, ch\u1ea5t chuy\u1ec3n h\u00f3a c\u00f3 n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh 80-100 ng\/mL trong v\u00f2ng 2,5-4 gi\u1edd. Li\u1ec1u 20 mg t\u1ea1o n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh ebastin kho\u1ea3ng 2,8 ng\/mL v\u00e0 carebastin kho\u1ea3ng 157 ng\/mL. Tr\u00ean 95% ebastin v\u00e0 carebastin c\u00f3 kh\u1ea3 n\u0103ng li\u00ean k\u1ebft protein huy\u1ebft t\u01b0\u01a1ng. D\u00f9ng Ebastin c\u00f9ng b\u1eefa \u0103n l\u00e0m t\u0103ng n\u1ed3ng \u0111\u1ed9 ch\u1ea5t chuy\u1ec3n h\u00f3a ho\u1ea1t t\u00ednh g\u1ea5p 1,6-2 l\u1ea7n, nh\u01b0ng kh\u00f4ng \u1ea3nh h\u01b0\u1edfng \u0111\u1ebfn Cmax hay hi\u1ec7u qu\u1ea3 \u0111i\u1ec1u tr\u1ecb.<\/p>\n

Chuy\u1ec3n h\u00f3a: Ebastin \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a qua gan ho\u00e0n to\u00e0n th\u00e0nh carebastin c\u00f3 ho\u1ea1t t\u00ednh.<\/p>\n

Th\u1ea3i tr\u1eeb: Th\u1eddi gian b\u00e1n th\u1ea3i c\u1ee7a carebastin kho\u1ea3ng 15-19 gi\u1edd, kho\u1ea3ng 66% \u0111\u01b0\u1ee3c \u0111\u00e0o th\u1ea3i qua n\u01b0\u1edbc ti\u1ec3u d\u01b0\u1edbi d\u1ea1ng li\u00ean h\u1ee3p.<\/p>\n

Thu\u1ed1c Atirin Suspension \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

Thu\u1ed1c Atirin Suspension<\/strong> \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong c\u00e1c tr\u01b0\u1eddng h\u1ee3p:<\/p>\n