{"id":125999,"date":"2025-07-04T16:57:20","date_gmt":"2025-07-04T09:57:20","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=125999"},"modified":"2025-12-23T10:24:32","modified_gmt":"2025-12-23T03:24:32","slug":"huether-25","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/huether-25\/","title":{"rendered":"Huether-25"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y,<\/strong> d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/strong><\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c<\/strong> Huether-25 \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi C\u00f4ng ty c\u1ed5 ph\u1ea7n d\u01b0\u1ee3c ph\u1ea9m \u0110\u1ea1t Vi Ph\u00fa (Davipharm), c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 893110593524 (VD-28463-17).<\/strong><\/p>\n

Huether-25 l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

M\u1ed7i vi\u00ean Huether-25<\/strong> ch\u1ee9a 25mg ho\u1ea1t ch\u1ea5t Topiramate<\/strong>. Topiramate l\u00e0 th\u00e0nh ph\u1ea7n d\u01b0\u1ee3c l\u00fd ch\u00ednh ch\u1ecbu tr\u00e1ch nhi\u1ec7m cho c\u00e1c t\u00e1c d\u1ee5ng \u0111i\u1ec1u tr\u1ecb c\u1ee7a thu\u1ed1c.<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: 893110593524 (VD-28463-17)<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 6 v\u1ec9 x 10 vi\u00ean<\/p>\n

Xu\u1ea5t x\u1ee9: Vi\u1ec7t Nam<\/p>\n

\"Huether-25
Huether-25 \u0111i\u1ec1u tr\u1ecb \u0111\u1ed9ng kinh<\/figcaption><\/figure>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Huether-25<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

Topiramate t\u00e1c \u0111\u1ed9ng th\u00f4ng qua nhi\u1ec1u c\u01a1 ch\u1ebf kh\u00e1c nhau tr\u00ean h\u1ec7 th\u1ea7n kinh trung \u01b0\u01a1ng:<\/p>\n

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  • Ch\u1eb9n k\u00eanh natri ph\u1ee5 thu\u1ed9c \u0111i\u1ec7n th\u1ebf: \u1ee8c ch\u1ebf c\u00e1c k\u00eanh natri, gi\u00fap \u1ed5n \u0111\u1ecbnh m\u00e0ng t\u1ebf b\u00e0o th\u1ea7n kinh v\u00e0 ng\u0103n ch\u1eb7n s\u1ef1 ph\u00e1t sinh \u0111i\u1ec7n th\u1ebf ho\u1ea1t \u0111\u1ed9ng l\u1eb7p l\u1ea1i nhanh ch\u00f3ng, gi\u1ea3m h\u01b0ng ph\u1ea5n qu\u00e1 m\u1ee9c c\u1ee7a t\u1ebf b\u00e0o th\u1ea7n kinh.<\/li>\n
  • T\u0103ng c\u01b0\u1eddng ho\u1ea1t \u0111\u1ed9ng GABA: T\u0103ng c\u01b0\u1eddng ho\u1ea1t \u0111\u1ed9ng c\u1ee7a GABA, m\u1ed9t ch\u1ea5t d\u1eabn truy\u1ec1n th\u1ea7n kinh \u1ee9c ch\u1ebf, th\u00f4ng qua vi\u1ec7c \u0111i\u1ec1u bi\u1ebfn c\u00e1c th\u1ee5 th\u1ec3 GABA-A, l\u00e0m t\u0103ng d\u00f2ng ion clorua v\u00e0o t\u1ebf b\u00e0o th\u1ea7n kinh.<\/li>\n
  • \u0110\u1ed1i kh\u00e1ng th\u1ee5 th\u1ec3 AMPA\/kainate c\u1ee7a glutamat: Ch\u1eb7n c\u00e1c th\u1ee5 th\u1ec3 AMPA v\u00e0 kainate, l\u00e0m gi\u1ea3m t\u00edn hi\u1ec7u k\u00edch th\u00edch trong n\u00e3o.<\/li>\n
  • \u1ee8c ch\u1ebf enzym carbonic anhydrase: \u1ee8c ch\u1ebf ch\u1ecdn l\u1ecdc c\u00e1c d\u1ea1ng enzym carbonic anhydrase, c\u00f3 th\u1ec3 g\u00f3p ph\u1ea7n v\u00e0o t\u00e1c d\u1ee5ng ch\u1ed1ng co gi\u1eadt.<\/li>\n
  • \u1ee8c ch\u1ebf k\u00eanh canxi lo\u1ea1i L: Gi\u1ea3m d\u00f2ng ion canxi v\u00e0o t\u1ebf b\u00e0o th\u1ea7n kinh, gi\u1ea3m t\u00ednh h\u01b0ng ph\u1ea5n.<\/li>\n<\/ul>\n

    \u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n
      \n
    • H\u1ea5p thu: Topiramate \u0111\u01b0\u1ee3c h\u1ea5p thu t\u1ed1t t\u1eeb \u0111\u01b0\u1eddng ti\u00eau h\u00f3a (>80% sinh kh\u1ea3 d\u1ee5ng). N\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng \u0111\u1ea1t \u0111\u01b0\u1ee3c trong kho\u1ea3ng 2-3 gi\u1edd.<\/li>\n
    • Ph\u00e2n b\u1ed1: T\u1ef7 l\u1ec7 g\u1eafn k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng th\u1ea5p (15% \u0111\u1ebfn 41% ho\u1eb7c 9% \u0111\u1ebfn 17% ), gi\u1ea3m thi\u1ec3u nguy c\u01a1 t\u01b0\u01a1ng t\u00e1c thu\u1ed1c do c\u1ea1nh tranh v\u1ecb tr\u00ed g\u1eafn k\u1ebft protein. Th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 l\u00e0 0.6-0.8 L\/kg.<\/li>\n
    • Chuy\u1ec3n h\u00f3a: Kho\u1ea3ng 20% Topiramate \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a \u1edf gan, t\u1ef7 l\u1ec7 n\u00e0y c\u00f3 th\u1ec3 t\u0103ng l\u00ean \u0111\u1ebfn 50% khi c\u00f3 m\u1eb7t c\u00e1c thu\u1ed1c g\u00e2y c\u1ea3m \u1ee9ng enzym.<\/li>\n
    • Th\u1ea3i tr\u1eeb: Topiramate th\u1ea3i tr\u1eeb ch\u1ee7 y\u1ebfu qua th\u1eadn, c\u1ea3 d\u01b0\u1edbi d\u1ea1ng kh\u00f4ng \u0111\u1ed5i v\u00e0 d\u1ea1ng ch\u1ea5t chuy\u1ec3n h\u00f3a. Th\u1eddi gian b\u00e1n th\u1ea3i trung b\u00ecnh trong huy\u1ebft t\u01b0\u01a1ng kho\u1ea3ng 21 gi\u1edd.<\/li>\n<\/ul>\n

      Thu\u1ed1c Huether-25 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n
        \n
      • \u0110i\u1ec1u tr\u1ecb \u0111\u1ed9ng kinh:\n
          \n
        • \u0110\u01a1n tr\u1ecb li\u1ec7u ban \u0111\u1ea7u cho b\u1ec7nh nh\u00e2n t\u1eeb 2 tu\u1ed5i tr\u1edf l\u00ean c\u00f3 c\u00e1c c\u01a1n \u0111\u1ed9ng kinh kh\u1edfi ph\u00e1t c\u1ee5c b\u1ed9 ho\u1eb7c co c\u1ee9ng-co gi\u1eadt to\u00e0n th\u00e2n nguy\u00ean ph\u00e1t.<\/li>\n
        • Li\u1ec7u ph\u00e1p h\u1ed7 tr\u1ee3 cho ng\u01b0\u1eddi l\u1edbn v\u00e0 tr\u1ebb em t\u1eeb 2 \u0111\u1ebfn 16 tu\u1ed5i c\u00f3 c\u00e1c c\u01a1n \u0111\u1ed9ng kinh kh\u1edfi ph\u00e1t c\u1ee5c b\u1ed9 ho\u1eb7c co c\u1ee9ng-co gi\u1eadt to\u00e0n th\u00e2n nguy\u00ean ph\u00e1t.<\/li>\n
        • Li\u1ec7u ph\u00e1p h\u1ed7 tr\u1ee3 cho b\u1ec7nh nh\u00e2n t\u1eeb 2 tu\u1ed5i tr\u1edf l\u00ean b\u1ecb c\u00e1c c\u01a1n \u0111\u1ed9ng kinh li\u00ean quan \u0111\u1ebfn h\u1ed9i ch\u1ee9ng Lennox-Gastaut.<\/li>\n<\/ul>\n<\/li>\n
        • D\u1ef1 ph\u00f2ng \u0111au n\u1eeda \u0111\u1ea7u: \u0110\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh \u0111\u1ec3 d\u1ef1 ph\u00f2ng \u0111au n\u1eeda \u0111\u1ea7u \u1edf ng\u01b0\u1eddi l\u1edbn v\u00e0 tr\u1ebb em t\u1eeb 12 tu\u1ed5i tr\u1edf l\u00ean. C\u1ea7n l\u01b0u \u00fd thu\u1ed1c ch\u1ec9 c\u00f3 t\u00e1c d\u1ee5ng d\u1ef1 ph\u00f2ng ho\u1eb7c gi\u1ea3m s\u1ed1 l\u01b0\u1ee3ng c\u01a1n \u0111au n\u1eeda \u0111\u1ea7u, kh\u00f4ng \u0111i\u1ec1u tr\u1ecb c\u01a1n \u0111au \u0111\u1ea7u \u0111\u00e3 kh\u1edfi ph\u00e1t.<\/li>\n<\/ul>\n

          Li\u1ec1u d\u00f9ng c\u1ee7a thu\u1ed1c Huether-25<\/h2>\n\n\n\n\n\n\n\n\n
          Ch\u1ec9 \u0111\u1ecbnh<\/td>\n\u0110\u1ed1i t\u01b0\u1ee3ng<\/td>\nLi\u1ec1u kh\u1edfi \u0111\u1ea7u<\/td>\nT\u1ed1c \u0111\u1ed9 d\u00f2 li\u1ec1u<\/td>\nLi\u1ec1u m\u1ee5c ti\u00eau\/duy tr\u00ec<\/td>\nLi\u1ec1u t\u1ed1i \u0111a khuy\u1ebfn c\u00e1o<\/td>\n<\/tr>\n
          \u0110\u01a1n tr\u1ecb li\u1ec7u \u0111\u1ed9ng kinh<\/td>\nNg\u01b0\u1eddi l\u1edbn<\/td>\n25 mg\/ng\u00e0y (u\u1ed1ng bu\u1ed5i t\u1ed1i) trong 1 tu\u1ea7n<\/td>\nT\u0103ng 25-50 mg\/ng\u00e0y m\u1ed7i 1-2 tu\u1ea7n, chia 2 l\u1ea7n<\/td>\nKho\u1ea3ng 400 mg\/ng\u00e0y, chia 2 l\u1ea7n<\/td>\n1.000 mg\/ng\u00e0y (m\u1ed9t s\u1ed1 b\u1ec7nh nh\u00e2n kh\u00e1ng thu\u1ed1c dung n\u1ea1p)<\/td>\n<\/tr>\n
          \u0110i\u1ec1u tr\u1ecb h\u1ed7 tr\u1ee3 \u0111\u1ed9ng kinh<\/td>\nTr\u1ebb em (\u2265 2 tu\u1ed5i)<\/td>\n25 mg\/ng\u00e0y (u\u1ed1ng bu\u1ed5i t\u1ed1i) trong 1 tu\u1ea7n (ho\u1eb7c 1-3 mg\/kg\/ng\u00e0y)<\/td>\nT\u0103ng 1-3 mg\/kg\/ng\u00e0y m\u1ed7i 1-2 tu\u1ea7n, chia 2 l\u1ea7n<\/td>\nD\u00f2 li\u1ec1u trong 5-7 tu\u1ea7n \u0111\u1ec3 \u0111\u1ea1t li\u1ec1u duy tr\u00ec d\u1ef1a tr\u00ean c\u00e2n n\u1eb7ng<\/td>\n30 mg\/kg\/ng\u00e0y (t\u1ed5ng li\u1ec1u kh\u00f4ng qu\u00e1 400 mg\/ng\u00e0y)<\/td>\n<\/tr>\n
          Ng\u01b0\u1eddi l\u1edbn<\/td>\n25-50 mg\/ng\u00e0y (u\u1ed1ng bu\u1ed5i t\u1ed1i) trong 1 tu\u1ea7n<\/td>\nT\u0103ng 25-50 mg\/ng\u00e0y m\u1ed7i 1-2 tu\u1ea7n, chia 2 l\u1ea7n<\/td>\nKho\u1ea3ng 200-400 mg\/ng\u00e0y, chia 2 l\u1ea7n<\/td>\n500 mg\/ng\u00e0y<\/td>\n<\/tr>\n
          Tr\u1ebb em (\u2265 2 tu\u1ed5i)<\/td>\n25 mg\/ng\u00e0y (u\u1ed1ng bu\u1ed5i t\u1ed1i) trong 1 tu\u1ea7n (ho\u1eb7c 1-3 mg\/kg\/ng\u00e0y)<\/td>\nT\u0103ng 1-3 mg\/kg\/ng\u00e0y m\u1ed7i 1-2 tu\u1ea7n, chia 2 l\u1ea7n<\/td>\nKho\u1ea3ng 5-9 mg\/kg\/ng\u00e0y, chia 2 l\u1ea7n<\/td>\nT\u1ed5ng li\u1ec1u kh\u00f4ng qu\u00e1 400 mg\/ng\u00e0y<\/td>\n<\/tr>\n
          D\u1ef1 ph\u00f2ng \u0111au n\u1eeda \u0111\u1ea7u<\/td>\nNg\u01b0\u1eddi l\u1edbn v\u00e0 tr\u1ebb em (\u2265 12 tu\u1ed5i)<\/td>\n25 mg\/ng\u00e0y (u\u1ed1ng bu\u1ed5i t\u1ed1i) trong 1 tu\u1ea7n<\/td>\nT\u0103ng 25 mg\/ng\u00e0y m\u1ed7i tu\u1ea7n<\/td>\n100 mg\/ng\u00e0y, chia 2 l\u1ea7n<\/td>\n200 mg\/ng\u00e0y (c\u1ea7n th\u1eadn tr\u1ecdng do t\u0103ng t\u00e1c d\u1ee5ng ph\u1ee5)<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n

          C\u00e1ch d\u00f9ng c\u1ee7a thu\u1ed1c Huether-25<\/h2>\n