{"id":125906,"date":"2025-07-04T14:07:02","date_gmt":"2025-07-04T07:07:02","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=125906"},"modified":"2025-07-24T11:46:40","modified_gmt":"2025-07-24T04:46:40","slug":"etoricoxib-60-khapharco","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/etoricoxib-60-khapharco\/","title":{"rendered":"Etoricoxib 60 Khapharco"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y, d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n thu\u1ed1c Etoricoxib 60 \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi C\u00f4ng ty c\u1ed5 ph\u1ea7n d\u01b0\u1ee3c ph\u1ea9m Kh\u00e1nh H\u00f2a c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 893110287523 (S\u0110K c\u0169: VD-27915-17)<\/strong><\/p>\n

Etoricoxib 60 l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

Trong m\u1ed7i vi\u00ean u\u1ed1ng Etoricoxib 60<\/strong> c\u00f3 ch\u1ee9a:<\/p>\n

Etoricoxib\u2026\u2026\u2026\u2026\u2026\u2026..60mg<\/p>\n

D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: 893110287523 (S\u0110K c\u0169: VD-27915-17)<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 1 chai 500 vi\u00ean<\/p>\n

Xu\u1ea5t x\u1ee9: Vi\u1ec7t Nam<\/p>\n

H\u1ea1n s\u1eed d\u1ee5ng: 36 th\u00e1ng<\/p>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Etoricoxib 60<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

Etoricoxib l\u00e0 thu\u1ed1c thu\u1ed9c nh\u00f3m \u1ee9c ch\u1ebf ch\u1ecdn l\u1ecdc enzym cyclooxygenase-2 (COX-2) \u2013 m\u1ed9t enzym th\u00fac \u0111\u1ea9y qu\u00e1 tr\u00ecnh t\u1ed5ng h\u1ee3p prostaglandin t\u1ea1i v\u1ecb tr\u00ed vi\u00eam. B\u1eb1ng c\u00e1ch \u1ee9c ch\u1ebf COX-2, thu\u1ed1c gi\u00fap l\u00e0m gi\u1ea3m c\u00e1c bi\u1ec3u hi\u1ec7n s\u01b0ng, n\u00f3ng, \u0111\u1ecf, \u0111au do vi\u00eam. \u0110\u1eb7c bi\u1ec7t, Etoricoxib kh\u00f4ng \u1ea3nh h\u01b0\u1edfng \u0111\u00e1ng k\u1ec3 t\u1edbi COX-1 \u2013 enzym c\u00f3 vai tr\u00f2 b\u1ea3o v\u1ec7 ni\u00eam m\u1ea1c d\u1ea1 d\u00e0y v\u00e0 ch\u1ee9c n\u0103ng ti\u1ec3u c\u1ea7u \u2013 do \u0111\u00f3 h\u1ea1n ch\u1ebf \u0111\u01b0\u1ee3c t\u00e1c d\u1ee5ng ph\u1ee5 tr\u00ean ti\u00eau h\u00f3a v\u00e0 \u0111\u00f4ng m\u00e1u so v\u1edbi NSAID truy\u1ec1n th\u1ed1ng.<\/p>\n

\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h2>\n

H\u1ea5p thu<\/h3>\n

Etoricoxib \u0111\u01b0\u1ee3c h\u1ea5p thu nhanh ch\u00f3ng qua \u0111\u01b0\u1eddng ti\u00eau h\u00f3a khi d\u00f9ng \u0111\u01b0\u1eddng u\u1ed1ng, v\u1edbi sinh kh\u1ea3 d\u1ee5ng g\u1ea7n nh\u01b0 ho\u00e0n to\u00e0n. \u1ede tr\u1ea1ng th\u00e1i \u1ed5n \u0111\u1ecbnh sau khi d\u00f9ng li\u1ec1u 120 mg, n\u1ed3ng \u0111\u1ed9 \u0111\u1ec9nh trong huy\u1ebft t\u01b0\u01a1ng \u0111\u1ea1t \u0111\u01b0\u1ee3c sau kho\u1ea3ng 1 gi\u1edd. T\u1ed5ng di\u1ec7n t\u00edch d\u01b0\u1edbi \u0111\u01b0\u1eddng cong (AUC) cho th\u1ea5y kh\u1ea3 n\u0103ng h\u1ea5p thu \u1ed5n \u0111\u1ecbnh v\u00e0 tuy\u1ebfn t\u00ednh trong ph\u1ea1m vi li\u1ec1u \u0111i\u1ec1u tr\u1ecb. Vi\u1ec7c d\u00f9ng thu\u1ed1c k\u00e8m b\u1eefa \u0103n gi\u00e0u ch\u1ea5t b\u00e9o c\u00f3 th\u1ec3 l\u00e0m ch\u1eadm t\u1ed1c \u0111\u1ed9 h\u1ea5p thu nh\u01b0ng kh\u00f4ng \u1ea3nh h\u01b0\u1edfng \u0111\u1ebfn m\u1ee9c \u0111\u1ed9 h\u1ea5p thu to\u00e0n ph\u1ea7n, do \u0111\u00f3 kh\u00f4ng c\u1ea7n \u0111i\u1ec1u ch\u1ec9nh theo b\u1eefa \u0103n.<\/p>\n

Ph\u00e2n b\u1ed1<\/h3>\n

Etoricoxib g\u1eafn k\u1ebft m\u1ea1nh v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng ng\u01b0\u1eddi (kho\u1ea3ng 92%) \u1edf n\u1ed3ng \u0111\u1ed9 tr\u1ecb li\u1ec7u. Th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 bi\u1ec3u ki\u1ebfn khi \u0111\u1ea1t tr\u1ea1ng th\u00e1i \u1ed5n \u0111\u1ecbnh v\u00e0o kho\u1ea3ng 120 l\u00edt, cho th\u1ea5y thu\u1ed1c ph\u00e2n b\u1ed1 r\u1ed9ng r\u00e3i v\u00e0o c\u00e1c m\u00f4. D\u1eef li\u1ec7u tr\u00ean \u0111\u1ed9ng v\u1eadt c\u0169ng ghi nh\u1eadn etoricoxib c\u00f3 kh\u1ea3 n\u0103ng v\u01b0\u1ee3t qua h\u00e0ng r\u00e0o m\u00e1u n\u00e3o v\u00e0 nhau thai.<\/p>\n

Chuy\u1ec3n h\u00f3a<\/h3>\n

Thu\u1ed1c \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a g\u1ea7n nh\u01b0 ho\u00e0n to\u00e0n t\u1ea1i gan, v\u1edbi ch\u01b0a \u0111\u1ebfn 1% l\u01b0\u1ee3ng thu\u1ed1c nguy\u00ean v\u1eb9n \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y trong n\u01b0\u1edbc ti\u1ec3u. Qu\u00e1 tr\u00ecnh chuy\u1ec3n h\u00f3a ch\u1ee7 y\u1ebfu x\u1ea3y ra th\u00f4ng qua c\u00e1c enzyme cytochrome P450, trong \u0111\u00f3 vai tr\u00f2 ch\u00ednh thu\u1ed9c v\u1ec1 CYP3A4. M\u1ed9t s\u1ed1 isoenzyme kh\u00e1c nh\u01b0 CYP2D6, CYP2C9, CYP1A2 v\u00e0 CYP2C19 c\u0169ng tham gia, nh\u01b0ng m\u1ee9c \u0111\u1ed9 \u1ea3nh h\u01b0\u1edfng ch\u01b0a \u0111\u01b0\u1ee3c x\u00e1c \u0111\u1ecbnh r\u00f5. C\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a ch\u00ednh c\u1ee7a etoricoxib kh\u00f4ng c\u00f2n ho\u1ea1t t\u00ednh ho\u1eb7c ch\u1ec9 c\u00f2n ho\u1ea1t t\u00ednh y\u1ebfu \u0111\u1ed1i v\u1edbi COX-2 v\u00e0 kh\u00f4ng \u1ea3nh h\u01b0\u1edfng \u0111\u1ebfn COX-1.<\/p>\n

Th\u1ea3i tr\u1eeb<\/h3>\n

Sau khi d\u00f9ng m\u1ed9t li\u1ec1u c\u00f3 g\u1eafn \u0111\u1ed3ng v\u1ecb ph\u00f3ng x\u1ea1, ph\u1ea7n l\u1edbn ho\u1ea1t ch\u1ea5t \u0111\u01b0\u1ee3c \u0111\u00e0o th\u1ea3i qua n\u01b0\u1edbc ti\u1ec3u (kho\u1ea3ng 70%) v\u00e0 ph\u00e2n (20%), ch\u1ee7 y\u1ebfu d\u01b0\u1edbi d\u1ea1ng \u0111\u00e3 chuy\u1ec3n h\u00f3a. Ch\u1ec9 d\u01b0\u1edbi 2% thu\u1ed1c \u0111\u01b0\u1ee3c b\u00e0i ti\u1ebft \u1edf d\u1ea1ng c\u00f2n nguy\u00ean. Etoricoxib c\u00f3 th\u1eddi gian b\u00e1n h\u1ee7y d\u00e0i, v\u00e0o kho\u1ea3ng 22 gi\u1edd, v\u1edbi tr\u1ea1ng th\u00e1i \u1ed5n \u0111\u1ecbnh \u0111\u1ea1t \u0111\u01b0\u1ee3c sau kho\u1ea3ng m\u1ed9t tu\u1ea7n d\u00f9ng thu\u1ed1c \u0111\u1ec1u \u0111\u1eb7n. \u0110\u1ed9 thanh th\u1ea3i to\u00e0n th\u00e2n c\u1ee7a thu\u1ed1c v\u00e0o kho\u1ea3ng 50 mL\/ph\u00fat.<\/p>\n

Thu\u1ed1c Etoricoxib 60 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n