{"id":120326,"date":"2025-05-26T16:53:55","date_gmt":"2025-05-26T09:53:55","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=120326"},"modified":"2025-07-24T13:13:27","modified_gmt":"2025-07-24T06:13:27","slug":"fripitor-10","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/fripitor-10\/","title":{"rendered":"Fripitor 10"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y, d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/a> s\u1ebd gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c Fripitor 10<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi C\u00f4ng ty c\u1ed5 ph\u1ea7n D\u01b0\u1ee3c ph\u1ea9m Fremed, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VD-36008-22.<\/strong><\/p>\n

Fripitor 10 l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

M\u1ed7i vi\u00ean n\u00e9n bao phim thu\u1ed1c Fripitor 10<\/strong> ch\u1ee9a:<\/p>\n

    \n
  • Atorvastatin calcium (t\u01b0\u01a1ng \u0111\u01b0\u01a1ng 10mg atorvastatin) 10,34mg<\/li>\n
  • T\u00e1 d\u01b0\u1ee3c v\u1eeba \u0111\u1ee7.<\/li>\n<\/ul>\n

    D\u1ea1ng b\u00e0o ch\u1ebf: Vi\u00ean n\u00e9n bao phim.<\/p>\n

    \"Fripitor
    Fripitor 10 \u0111i\u1ec1u tr\u1ecb t\u0103ng cholesterol m\u00e1u<\/figcaption><\/figure>\n

    Tr\u00ecnh b\u00e0y<\/h3>\n

    S\u0110K: VD-36008-22<\/p>\n

    Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 3 v\u1ec9 x 10 vi\u00ean<\/p>\n

    Xu\u1ea5t x\u1ee9: Vi\u1ec7t Nam<\/p>\n

    H\u1ea1n s\u1eed d\u1ee5ng: 24 th\u00e1ng<\/p>\n

    T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Fripitor 10<\/h2>\n

    C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

    Atorvastatin l\u00e0 m\u1ed9t ch\u1ea5t \u1ee9c ch\u1ebf ch\u1ecdn l\u1ecdc v\u00e0 c\u1ea1nh tranh enzyme HMG-CoA reductase – enzyme tham gia b\u01b0\u1edbc \u0111\u1ea7u trong qu\u00e1 tr\u00ecnh t\u1ed5ng h\u1ee3p cholesterol t\u1ea1i gan.<\/p>\n

    Atorvastatin gi\u00fap gi\u1ea3m n\u1ed3ng \u0111\u1ed9 cholesterol trong m\u00e1u b\u1eb1ng c\u00e1ch h\u1ea1n ch\u1ebf s\u1ea3n xu\u1ea5t cholesterol t\u1ea1i gan v\u00e0 t\u0103ng l\u01b0\u1ee3ng th\u1ee5 th\u1ec3 LDL \u1edf b\u1ec1 m\u1eb7t t\u1ebf b\u00e0o gan, qua \u0111\u00f3 t\u0103ng c\u01b0\u1eddng h\u1ea5p thu v\u00e0 ph\u00e2n gi\u1ea3i LDL. Thu\u1ed1c l\u00e0m gi\u1ea3m c\u1ea3 s\u1ef1 s\u1ea3n sinh v\u00e0 s\u1ed1 l\u01b0\u1ee3ng ph\u00e2n t\u1eed LDL, \u0111\u1ed3ng th\u1eddi c\u1ea3i thi\u1ec7n ch\u1ea5t l\u01b0\u1ee3ng c\u1ee7a ch\u00fang trong tu\u1ea7n ho\u00e0n.<\/p>\n

    \u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

    H\u1ea5p thu: Atorvastatin \u0111\u01b0\u1ee3c h\u1ea5p thu nhanh sau khi u\u1ed1ng, \u0111\u1ea1t n\u1ed3ng \u0111\u1ed9 cao nh\u1ea5t trong huy\u1ebft t\u01b0\u01a1ng sau kho\u1ea3ng 1-2 gi\u1edd. Sinh kh\u1ea3 d\u1ee5ng tuy\u1ec7t \u0111\u1ed1i c\u1ee7a atorvastatin v\u00e0o kho\u1ea3ng 12%, trong khi ho\u1ea1t t\u00ednh \u1ee9c ch\u1ebf enzym HMG-CoA reductase c\u00f3 sinh kh\u1ea3 d\u1ee5ng kho\u1ea3ng 30%. S\u1ef1 h\u1ea5p thu th\u1ea5p ch\u1ee7 y\u1ebfu do thu\u1ed1c b\u1ecb chuy\u1ec3n h\u00f3a m\u1ed9t ph\u1ea7n t\u1ea1i ni\u00eam m\u1ea1c ru\u1ed9t v\u00e0 gan tr\u01b0\u1edbc khi v\u00e0o v\u00f2ng tu\u1ea7n ho\u00e0n chung.<\/p>\n

    Ph\u00e2n b\u1ed1: Th\u1ec3 t\u00edch ph\u00e2n b\u1ed1 c\u1ee7a thu\u1ed1c v\u00e0o kho\u1ea3ng 381 l\u00edt, v\u1edbi h\u01a1n 98% li\u00ean k\u1ebft v\u1edbi protein huy\u1ebft t\u01b0\u01a1ng. Nghi\u00ean c\u1ee9u tr\u00ean \u0111\u1ed9ng v\u1eadt cho th\u1ea5y thu\u1ed1c c\u00f3 th\u1ec3 b\u00e0i ti\u1ebft v\u00e0o s\u1eefa.<\/p>\n

    Chuy\u1ec3n h\u00f3a: Atorvastatin ch\u1ee7 y\u1ebfu \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a t\u1ea1i gan nh\u1edd enzym CYP3A4, t\u1ea1o th\u00e0nh c\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a hydroxyl h\u00f3a t\u1ea1i v\u1ecb tr\u00ed ortho v\u00e0 para, c\u0169ng nh\u01b0 c\u00e1c s\u1ea3n ph\u1ea9m oxy h\u00f3a \u1edf v\u1ecb tr\u00ed beta.<\/p>\n

    Th\u1ea3i tr\u1eeb: Thu\u1ed1c v\u00e0 c\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a \u0111\u01b0\u1ee3c \u0111\u00e0o th\u1ea3i ch\u1ee7 y\u1ebfu qua m\u1eadt, sau khi chuy\u1ec3n h\u00f3a t\u1ea1i gan ho\u1eb7c ngo\u00e0i gan, nh\u01b0ng kh\u00f4ng c\u00f3 chu tr\u00ecnh gan-ru\u1ed9t. Th\u1eddi gian b\u00e1n th\u1ea3i c\u1ee7a atorvastatin kho\u1ea3ng 14 gi\u1edd, trong khi t\u00e1c d\u1ee5ng \u1ee9c ch\u1ebf enzym HMG-CoA reductase k\u00e9o d\u00e0i h\u01a1n (20-30 gi\u1edd), nh\u1edd c\u00e1c ch\u1ea5t chuy\u1ec3n h\u00f3a v\u1eabn c\u00f2n ho\u1ea1t t\u00ednh. D\u01b0\u1edbi 2% li\u1ec1u u\u1ed1ng \u0111\u01b0\u1ee3c b\u00e0i ti\u1ebft qua n\u01b0\u1edbc ti\u1ec3u.<\/p>\n

    Thu\u1ed1c Fripitor 10 \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

    Fripitor 10\u00a0\u0111\u01b0\u1ee3c d\u00f9ng ph\u1ed1i h\u1ee3p v\u1edbi ch\u1ebf \u0111\u1ed9 \u0103n \u0111\u1ec3 gi\u1ea3m cholesterol to\u00e0n ph\u1ea7n, LDL-C, apolipoprotein B v\u00e0 triglycerid \u1edf ng\u01b0\u1eddi t\u1eeb 10 tu\u1ed5i tr\u1edf l\u00ean m\u1eafc t\u0103ng cholesterol m\u00e1u nguy\u00ean ph\u00e1t (bao g\u1ed3m c\u1ea3 d\u1ea1ng di truy\u1ec1n d\u1ecb h\u1ee3p t\u1eed) ho\u1eb7c r\u1ed1i lo\u1ea1n lipid m\u00e1u h\u1ed7n h\u1ee3p. Thu\u1ed1c \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh khi thay \u0111\u1ed5i l\u1ed1i s\u1ed1ng kh\u00f4ng mang l\u1ea1i hi\u1ec7u qu\u1ea3. Ngo\u00e0i ra, atorvastatin c\u00f2n d\u00f9ng cho ng\u01b0\u1eddi l\u1edbn b\u1ecb t\u0103ng cholesterol m\u00e1u di truy\u1ec1n \u0111\u1ed3ng h\u1ee3p t\u1eed v\u00e0 h\u1ed7 tr\u1ee3 ph\u00f2ng ng\u1eeba b\u1ec7nh tim m\u1ea1ch \u1edf ng\u01b0\u1eddi c\u00f3 nguy c\u01a1 cao.<\/p>\n

    Li\u1ec1u d\u00f9ng v\u00e0 c\u00e1ch s\u1eed d\u1ee5ng<\/h2>\n

    C\u00e1ch d\u00f9ng: U\u1ed1ng 1 l\u1ea7n\/ng\u00e0y, v\u00e0o b\u1ea5t k\u1ef3 th\u1eddi \u0111i\u1ec3m n\u00e0o, c\u00f3 th\u1ec3 c\u00f9ng ho\u1eb7c kh\u00f4ng c\u00f9ng th\u1ee9c \u0103n. B\u1ec7nh nh\u00e2n c\u1ea7n tu\u00e2n th\u1ee7 ch\u1ebf \u0111\u1ed9 \u0103n gi\u1ea3m cholesterol trong su\u1ed1t th\u1eddi gian \u0111i\u1ec1u tr\u1ecb.<\/p>\n

    Li\u1ec1u d\u00f9ng: B\u1eaft \u0111\u1ea7u v\u1edbi li\u1ec1u 10mg\/ng\u00e0y, \u0111i\u1ec1u ch\u1ec9nh li\u1ec1u theo m\u1ee9c LDL-C v\u00e0 \u0111\u00e1p \u1ee9ng c\u1ee7a c\u01a1 th\u1ec3 sau m\u1ed7i 4 tu\u1ea7n. Li\u1ec1u t\u1ed1i \u0111a l\u00e0 80mg\/ng\u00e0y.<\/p>\n

    Atorvastatin ch\u1ec9 n\u00ean \u0111\u01b0\u1ee3c k\u00ea \u0111\u01a1n cho tr\u1ebb b\u1edfi b\u00e1c s\u0129 c\u00f3 kinh nghi\u1ec7m \u0111i\u1ec1u tr\u1ecb r\u1ed1i lo\u1ea1n lipid m\u00e1u \u1edf tr\u1ebb nh\u1ecf. C\u1ea7n theo d\u00f5i \u0111\u1ecbnh k\u1ef3 \u0111\u1ec3 \u0111\u00e1nh gi\u00e1 hi\u1ec7u qu\u1ea3 \u0111i\u1ec1u tr\u1ecb. V\u1edbi tr\u1ebb tr\u00ean 10 tu\u1ed5i m\u1eafc t\u0103ng cholesterol m\u00e1u di truy\u1ec1n d\u1ecb h\u1ee3p t\u1eed, li\u1ec1u b\u1eaft \u0111\u1ea7u l\u00e0 10mg\/ng\u00e0y, c\u00f3 th\u1ec3 t\u0103ng \u0111\u1ebfn t\u1ed1i \u0111a 80mg\/ng\u00e0y t\u00f9y v\u00e0o m\u1ee9c \u0111\u1ed9 \u0111\u00e1p \u1ee9ng v\u00e0 kh\u1ea3 n\u0103ng dung n\u1ea1p. Li\u1ec1u n\u00ean \u0111\u01b0\u1ee3c \u0111i\u1ec1u ch\u1ec9nh theo m\u1ee5c ti\u00eau \u0111i\u1ec1u tr\u1ecb sau m\u1ed7i 4 tu\u1ea7n ho\u1eb7c l\u00e2u h\u01a1n.<\/p>\n

    Kh\u00f4ng s\u1eed d\u1ee5ng Fripitor 10 trong tr\u01b0\u1eddng h\u1ee3p n\u00e0o?<\/h2>\n

    Fripitor 10<\/strong>\u00a0kh\u00f4ng \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong c\u00e1c tr\u01b0\u1eddng h\u1ee3p:<\/p>\n