{"id":103102,"date":"2024-10-24T13:00:30","date_gmt":"2024-10-24T06:00:30","guid":{"rendered":"https:\/\/hmm88i.com\/drug\/?post_type=product&p=103102"},"modified":"2025-07-24T13:22:58","modified_gmt":"2025-07-24T06:22:58","slug":"nicardipine-aguettant-10mg-10ml","status":"publish","type":"product","link":"https:\/\/hmm88i.com\/drug\/nicardipine-aguettant-10mg-10ml\/","title":{"rendered":"Nicardipine Aguettant 10mg\/10ml"},"content":{"rendered":"

Trong b\u00e0i vi\u1ebft n\u00e0y, <\/b>d\u01b0\u1ee3c s\u0129 L\u01b0u V\u0103n Ho\u00e0ng<\/b><\/a> gi\u1edbi thi\u1ec7u \u0111\u1ebfn c\u00e1c b\u1ea1n s\u1ea3n ph\u1ea9m thu\u1ed1c Nicardipine Aguettant 10mg\/10ml<\/a> \u0111\u01b0\u1ee3c s\u1ea3n xu\u1ea5t b\u1edfi Laboratoire Aguettant, c\u00f3 s\u1ed1 \u0111\u0103ng k\u00fd l\u01b0u h\u00e0nh t\u1ea1i Vi\u1ec7t Nam l\u00e0 VN-19999-16.<\/b><\/p>\n

Thu\u1ed1c Nicardipine Aguettant 10mg\/10ml l\u00e0 thu\u1ed1c g\u00ec?<\/h2>\n

Th\u00e0nh ph\u1ea7n<\/h3>\n

M\u1ed7i \u1ed1ng thu\u1ed1c Nicardipine Aguettant 10mg\/10ml<\/b> bao g\u1ed3m c\u00e1c th\u00e0nh ph\u1ea7n:<\/p>\n\n\n\n\n\n
Ho\u1ea1t ch\u1ea5t<\/td>\nH\u00e0m l\u01b0\u1ee3ng<\/td>\n<\/tr>\n
Nicardipin Hydroclorid<\/td>\n10mg<\/td>\n<\/tr>\n
T\u00e1 d\u01b0\u1ee3c<\/td>\nv\u1eeba \u0111\u1ee7<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n

D\u1ea1ng b\u00e0o ch\u1ebf: Dung d\u1ecbch ti\u00eam truy\u1ec1n t\u0129nh m\u1ea1ch.<\/p>\n

Tr\u00ecnh b\u00e0y<\/h3>\n

S\u0110K: VN-19999-16.<\/p>\n

Quy c\u00e1ch \u0111\u00f3ng g\u00f3i: H\u1ed9p 10 \u1ed1ng x 10ml.<\/p>\n

Xu\u1ea5t x\u1ee9: Ph\u00e1p.<\/p>\n

T\u00e1c d\u1ee5ng c\u1ee7a thu\u1ed1c Nicardipine Aguettant 10mg\/10ml<\/h2>\n

C\u01a1 ch\u1ebf t\u00e1c d\u1ee5ng<\/h3>\n

Nicardipin l\u00e0 ch\u1ea5t ch\u1eb9n k\u00eanh canxi ch\u1eadm th\u1ebf h\u1ec7 2, \u0111\u01b0\u1ee3c x\u1ebfp v\u00e0o nh\u00f3m phenyl-dihydropyridin. Nicardipin c\u00f3 t\u00ednh ch\u1ecdn l\u1ecdc kh\u00e1 cao tr\u00ean k\u00eanh canxi type L \u1edf c\u01a1 tr\u01a1n c\u1ee7a m\u1ea1ch m\u00e1u h\u01a1n tr\u00ean c\u01a1 tim.<\/p>\n

V\u1edbi n\u1ed3ng \u0111\u1ed9 r\u1ea5t nh\u1ecf, thu\u1ed1c s\u1ebd ng\u0103n ch\u1eb7n d\u00f2ng canxi \u0111i v\u00e0o b\u00ean trong t\u1ebf b\u00e0o. T\u00e1c \u0111\u1ed9ng n\u00e0y s\u1ebd th\u1ec3 hi\u1ec7n r\u00f5 r\u00e0ng h\u01a1n tr\u00ean c\u01a1 tr\u01a1n \u0111\u1ed9ng m\u1ea1ch. \u0110i\u1ec1u n\u00e0y \u0111\u00e3 \u0111\u01b0\u1ee3c ph\u1ea3n \u00e1nh b\u1edfi c\u00e1c thay \u0111\u1ed5i nhanh ch\u00f3ng, quan tr\u1ecdng c\u1ee7a huy\u1ebft \u00e1p. S\u1ee9c co c\u01a1 tim kh\u00f4ng c\u00f3 bi\u1ebfn \u0111\u1ed5i \u0111\u00e1ng k\u1ec3.<\/p>\n

Khi d\u00f9ng v\u1edbi \u0111\u01b0\u1eddng to\u00e0n th\u00e2n, thu\u1ed1c n\u00e0y l\u00e0 m\u1ed9t ch\u1ea5t gi\u00e3n m\u1ea1ch kh\u00e1 m\u1ea1nh m\u1ebd v\u00e0 l\u00e0m gi\u1ea3m huy\u1ebft \u00e1p. Nh\u1ecbp tim t\u0103ng tho\u00e1ng qua, cung l\u01b0\u1ee3ng tim c\u0169ng t\u0103ng v\u00e0 k\u00e9o d\u00e0i theo do h\u1eadu t\u1ea3i gi\u1ea3m.<\/p>\n

\u0110\u1eb7c \u0111i\u1ec3m d\u01b0\u1ee3c \u0111\u1ed9ng h\u1ecdc<\/h3>\n

H\u1ea5p thu: Thu\u1ed1c Nicardipin \u0111\u01b0\u1ee3c ti\u00eam v\u00e0o c\u01a1 th\u1ec3 n\u00ean sinh kh\u1ea3 d\u1ee5ng g\u1ea7n nh\u01b0 ho\u00e0n to\u00e0n.<\/p>\n

Ph\u00e2n b\u1ed1: Nicardipin s\u1ebd g\u1eafn m\u1ea1nh v\u1edbi c\u00e1c protein huy\u1ebft t\u01b0\u01a1ng v\u1edbi d\u1ea3i n\u1ed3ng \u0111\u1ed9 kh\u00e1 r\u1ed9ng.<\/p>\n

Chuy\u1ec3n h\u00f3a: Thu\u1ed1c \u0111\u01b0\u1ee3c chuy\u1ec3n h\u00f3a nh\u1edd x\u00fac t\u00e1c t\u1eeb CYP450 3A4. Ch\u1ea5t chuy\u1ec3n h\u00f3a ch\u00ednh \u0111\u00e3 \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y t\u1ea1i n\u01b0\u1edbc ti\u1ec3u l\u00e0 glucuronid d\u1ea1ng hydroxy. Ch\u1ea5t n\u00e0y \u0111\u01b0\u1ee3c t\u1ea1o ra do qu\u00e1 tr\u00ecnh oxy h\u00f3a t\u00e1ch N-methylbenzen v\u00e0 v\u00f2ng pyridin.<\/p>\n

\u0110\u00e0o th\u1ea3i: Trong v\u00f2ng 96 ti\u1ebfng sau khi ti\u00eam t\u0129nh m\u1ea1ch, kho\u1ea3ng 49% thu\u1ed1c \u0111\u01b0\u1ee3c t\u00ecm th\u1ea5y \u1edf n\u01b0\u1edbc ti\u1ec3u, c\u00f2n 43% l\u00e0 \u1edf ph\u00e2n. Kh\u00f4ng t\u00ecm th\u1ea5y d\u1ea1ng ch\u01b0a bi\u1ebfn \u0111\u1ed5i \u1edf n\u01b0\u1edbc ti\u1ec3u. Sau khi ti\u00eam m\u1ed9t li\u1ec1u \u0111\u01b0\u1eddng t\u0129nh m\u1ea1ch, thu\u1ed1c s\u1ebd tr\u1ea3i qua 3 pha th\u1ea3i tr\u1eeb v\u1edbi c\u00e1c th\u1eddi gian b\u00e1n h\u1ee7y l\u00e0: alpha 6,4 ph\u00fat, beta 1,5 ti\u1ebfng v\u00e0 gamma 7,9 ti\u1ebfng.<\/p>\n

Thu\u1ed1c Nicardipine Aguettant 10mg\/10ml \u0111\u01b0\u1ee3c ch\u1ec9 \u0111\u1ecbnh trong b\u1ec7nh g\u00ec?<\/h2>\n

Thu\u1ed1c \u0111\u01b0\u1ee3c d\u00f9ng tr\u00ean b\u1ec7nh nh\u00e2n b\u1ecb t\u0103ng huy\u1ebft \u00e1p \u00e1c t\u00ednh \u1ea3nh h\u01b0\u1edfng t\u1edbi t\u00ednh m\u1ea1ng nh\u01b0:<\/p>\n